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3-phenyl-1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
5-cyclobutanecarbonyl-1'-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{[7-chloro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-4-methylbenzamide
1-methyl-4-[1-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)ethyl]piperazine
7-(cyclopropylmethyl)-2-(4-fluorobenzoyl)-2,7-diazaspiro[4.5]decan-6-one
3-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)propanamide
4-{2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}-N,N-dimethylpiperazine-1-carboxamide
2-(1H-pyrazol-1-ylmethyl)-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,4-oxazepane
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}furan-3-carboxamide
1-ethyl-6,7,8-trifluoro-3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,4-dihydroquinolin-4-one
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}[(4-methoxyphenyl)methyl](pyridin-4-ylmethyl)amine
8-[(5-methoxy-2-methyl-3-phenyl-1-benzofuran-6-yl)methyl]-1-(2-methoxyethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)acetamide
1-(2-{methyl[4-(trifluoromethyl)pyrimidin-2-yl]amino}ethyl)piperidin-2-one
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
6,8-dimethyl-2-{[4-(propan-2-yl)piperazin-1-yl]methyl}quinolin-4-ol
(1S,5R)-3-benzyl-6-[2-(4-fluorophenoxy)ethyl]-3,6-diazabicyclo[3.2.2]nonane
4-[4-({3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenyl]but-3-yn-1-ol
1-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
1-[1'-(4-hydroxybenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
2-(1H-imidazol-1-yl)-N-[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]acetamide
4-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyrimidin-2-amine
4-benzyl-3-{[1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}piperazin-2-one
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-2,3-dihydro-1-benzothiophene-2-carboxamide
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
4-[3-(dimethylamino)propyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3R,9aR)-8-benzoyl-3-[(1S)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3S,7S,8aS)-3-(1H-indol-3-ylmethyl)-7-{[(2-methylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-methyl-3-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole
N,4-dimethyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-1H-imidazole-5-carboxamide
1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-N-phenylpiperidin-3-amine
1-{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}piperidin-4-ol
2,3-dimethyl-6-{2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-({[(3R,4R)-4-(hydroxymethyl)-1-[5-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
6-[(2S,6S)-6-butyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-2-cyclopropyl-1,3-benzoxazole
2-cyclopropyl-5-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-4-methylpyrimidine
(1R,3S)-7-{2-amino-6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-3-ethoxy-7-azaspiro[3.5]nonan-1-ol
3-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}-5-methoxy-1H-indazole
(1S,5R)-3-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[1-(3-methylbutyl)-1H-pyrazol-4-yl]thiophene-2-carboxamide
N-methyl-1-(piperidin-3-ylmethyl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
5-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]oxane-4-carboxamide
2-butyl-4-methyl-N-(8-methylquinolin-5-yl)-3-oxopiperazine-1-carboxamide
N-cyclohexyl-3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-(prop-2-yn-1-yl)propanamide
N-(1-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide