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4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}benzamide
N-benzyl-1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-4-carboxamide
(1R,5R)-6-benzyl-3-(6-methyl-2-propylpyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonane
N,1,3-trimethyl-N-[2-methyl-3-(pyrrolidin-1-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1R,5R)-6-benzyl-3-(3-methoxy-4-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
2-(3-methoxyphenyl)-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)acetamide
2-(2-{[1-(2-methylpropyl)piperidin-4-yl]amino}ethyl)-1,2-dihydrophthalazin-1-one
N-[(3S,7S,8aS)-3-[(4-chlorophenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,4-dichlorobenzamide
1-{1-[(2-hydroxyphenyl)methyl]piperidin-4-yl}-N-(2-phenylethyl)piperidine-4-carboxamide
1-(1,4-dioxan-2-ylmethyl)-3-methyl-1,2-dihydroquinoxalin-2-one
1-(2-chlorophenyl)-3-{1-[1-(thian-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-[4-(4-methylphenyl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
1-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}-4-(methoxymethyl)piperidine
N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-1-(3-propanoylpiperidin-1-yl)propan-1-one
N-(1-cyclopropylethyl)-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
2-({5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}(propan-2-yl)amino)ethan-1-ol
[1-(1-benzylpiperidin-4-yl)-3-(2-phenylethyl)piperidin-3-yl]methanol
N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-3,4-dimethoxybenzamide
2-[(1-cyclobutanecarbonylpiperidin-4-yl)formamido]-3-(furan-2-yl)propanoic acid
(2E)-3-(3-fluorophenyl)-N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)prop-2-enamide
[(1-ethyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)(quinolin-4-ylmethyl)amine
N-{3-[6-amino-5-cyano-4-(cyclohex-3-en-1-yl)pyridin-2-yl]phenyl}acetamide
3-[4-(benzyloxy)piperidin-1-yl]-5-(3-fluorophenyl)-1,2,4-triazine
3-(diphenylmethyl)-5-(furan-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}propan-1-ol
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3-(1,2-oxazinan-2-yl)propanamide
1-(4-{[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
6-[3-oxo-3-(pyrrolidin-1-yl)propyl]-5,6-dihydro-1,6-naphthyridin-5-one
N-[2-methyl-1-(7-{[4-(methylsulfanyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]methanesulfonamide
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-ethyl-5-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
(1-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-2-phenylethyl)[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
(2E)-1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}-3-(thiophen-2-yl)prop-2-en-1-one
1-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
N-{[7-(2,3-dihydro-1-benzofuran-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
methyl 6-(1-methyl-1H-pyrazole-5-carbonyl)-2-[(2-phenylethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
ethyl 4-(cyclopropylmethyl)-1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylate
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-(5-hydroxypyrazine-2-carbonyl)-4-(2-methylphenoxy)piperidine-4-carboxylic acid
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-fluorophenyl)acetamide
1-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-3-[2-(prop-2-en-1-yloxy)phenyl]urea
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
2-(methylamino)-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]pyridine-4-carboxamide
4'-(cyclobutylmethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)cyclohexanamine
2-(2,4-dimethoxyphenyl)-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]acetic acid
3-[(cyclohex-3-en-1-ylmethyl)(propan-2-yl)amino]propanamide
(2S,4R)-4-(dimethylamino)-1-{[5-(4-ethoxyphenyl)furan-2-yl]methyl}pyrrolidine-2-carboxylic acid
2-methyl-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrido[2,3-d]pyrimidin-4-amine