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N-{[2-(1-ethyl-1H-indol-3-yl)-6-oxo-1,6-dihydropyrimidin-4-yl]methyl}acetamide
4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1λ6-thiomorpholine-1,1-dione
1-cycloheptyl-6-oxo-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
2-methyl-2-{2-[(3R)-3-methylpiperazin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}propanoic acid
1-(1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-3-yl)pyrrolidin-2-one
3-{5-[2-(azepan-1-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-cyclopropylpropanamide
methyl 3-{[(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl)carbamoyl}propanoate
(2S,4R)-4-amino-1-{3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propanoyl}-N-ethylpyrrolidine-2-carboxamide
(2S,6S)-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
N-cyclopropyl-1-[1-(thiophen-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N,6-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-(1,3-benzothiazol-2-yl)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)propanamide
3-benzoyl-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
2,5-dimethyl-N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)-1,3-thiazole-4-carboxamide
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-[(dimethylamino)methyl]-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}benzamide
N-[(6-hydroxypyrimidin-4-yl)methyl]-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
4-{4-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}quinazoline
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(1S,5R)-6-(5-ethyl-1,3-oxazole-4-carbonyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(3R,4R)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-ol
6-{1-methyl-5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}pyridine-2-carbonitrile
2-amino-N-benzyl-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(3-methylpyridin-2-yl)methyl]acetamide
8-benzyl-3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(1,2-oxazol-5-yl)-4-(3,4,5-trimethoxyphenyl)phenol
3-({methyl[(2-phenyl-1,3-thiazol-5-yl)methyl]amino}methyl)pyridin-2-amine
N-{[7-(4-chlorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-3-carboxamide
methyl 2-{1-[(3-fluorophenyl)carbamoyl]-6-azaspiro[2.5]octane-6-carbonyl}benzoate
4-(2,4-dioxoimidazolidin-1-yl)-N-[2-(N-methylmethanesulfonamido)ethyl]benzamide
(3S,4S)-4-cyclopropyl-1-{[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}pyrrolidine-3-carboxylic acid
2-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenol
1-(4-chloro-2,6-dimethylphenyl)-3-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]urea
N-[(3S,4R)-1-[3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
(1-{[1-(4-chloro-2-fluorobenzoyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
N-[2-(N-methylmethanesulfonamido)ethyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-N-methylpiperidine-2-carboxamide
N-[(2R,3R)-2-(prop-2-en-1-yloxy)-1'-(pyridine-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]cyclopropanecarboxamide
4-(1-butyl-1H-imidazol-2-yl)-1-(3-chloro-4-methoxybenzoyl)piperidine
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}acetamide
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-7-methyl-1-benzofuran-2-carboxamide
1-[(4,5-dimethylfuran-2-yl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
1-{5-[2-(azocan-1-yl)ethyl]-3-cyclopropyl-1H-1,2,4-triazol-1-yl}butan-2-ol
5-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]pyrrolidin-2-yl}-3-phenyl-1,2,4-oxadiazole
8-(2,2-diphenylethyl)-3-ethyl-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
(1S,3R)-N1,1,2,N2,N3,3-hexamethyl-N1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]cyclopentane-1,3-dicarboxamide
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,6-dimethylpyrimidin-4-amine
1-(2-methyl-1-benzofuran-5-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-ethyl-8-{[5-(oxan-2-yl)thiophen-2-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,6-dimethylpyridine-3-carboxamide