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3-[2-(azocan-1-yl)-2-oxoethyl]-4-[(2,3-dimethoxyphenyl)methyl]piperazin-2-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-1-methylcyclopropane-1-carboxamide
2-(2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamido)-N-methylacetamide
1-[1-(1-propylpiperidin-4-yl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
[(1-cyclopentylpiperidin-4-yl)methyl]({[2-(difluoromethoxy)phenyl]methyl})(oxolan-2-ylmethyl)amine
4-(2,5-dihydro-1H-pyrrole-2-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-[(diethylamino)methyl]-N-[(1-methylpyrrolidin-3-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
methyl 2-{[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinoline-1-carbonyl]amino}acetate
6-[4-(1,2,3,6-tetrahydropyridin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-9H-purine
1-[(4-methoxyphenyl)methyl]-4-[2-(oxolan-2-ylmethoxy)acetyl]piperazin-2-one
3-(3-fluorophenyl)-4-[(3-methyl-1-benzofuran-2-yl)methyl]piperazin-2-one
2-(1-phenylethyl)-1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazole
N-{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}-N-methylcyclohexanamine
2-(3-methylphenyl)-5-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]pyrimidin-4-ol
1-(3-fluorobenzoyl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(3-propyl-1H-pyrazole-5-carbonyl)-4-(1,3-thiazol-2-yl)piperazine
N-[1-({[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2H-1,3-benzodioxole-5-carboxamide
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
(3S,7S)-5-[3-(dimethylamino)pyrazin-2-yl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
5-ethyl-2-[4-(thian-4-yl)piperazin-1-yl]pyrimidine
8-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
[(3R,4R)-1-[1-(4-methylphenyl)piperidin-4-yl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
6-(cyclopropylmethoxy)-4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
1-[2-({1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-yl}amino)ethyl]imidazolidin-2-one
7-chloro-N-ethyl-4-hydroxy-N-[2-(1H-pyrazol-1-yl)ethyl]quinoline-3-carboxamide
8-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-1-(benzyloxy)-1,8-diazaspiro[4.5]decan-2-one
4-(1-{1-[(3-chloro-2,6-difluorophenyl)methyl]piperidin-4-yl}ethyl)morpholine
N-methyl-3-{1-[2-(4-methylphenoxy)acetyl]piperidin-3-yl}-N-[2-(pyridin-2-yl)ethyl]propanamide
3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}-N-(2-methylprop-2-en-1-yl)benzamide
(3R,4R)-4-amino-1-{2-[2-(3-methoxyphenyl)ethyl]benzoyl}piperidin-3-ol
3-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-ol
3-[benzyl(quinolin-4-ylmethyl)amino]-1λ6-thiolane-1,1-dione
N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
N-[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl]-2-[(1-methylpiperidin-4-yl)oxy]aniline
N-({5-[(4-methoxy-3-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
1-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}-4-(hydroxymethyl)azepan-4-ol
3-(1-methyl-1H-pyrazol-5-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}propanamide
N-methyl-3-(1H-pyrazol-1-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}benzamide
9-(2-methoxyethyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[(2-butyl-1H-imidazol-4-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
(3S,4S)-4-[({[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]piperidin-3-ol
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(pyrimidin-5-ylmethyl)pyrrolidine-3-carboxylic acid
7-(cyclopropylmethyl)-2-[3-(methylsulfanyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
(3S,7S)-5-[3-(methylcarbamoyl)pyridin-2-yl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
5-(3-fluorophenyl)-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1,2,4-triazin-3-amine
1-{4-[(butylamino)methyl]-2-methoxyphenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
3-phenyl-N-(2,2,2-trifluoroethyl)-1H-pyrazole-4-carboxamide
N-ethyl-5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-(pyridin-4-ylmethyl)pyridin-2-amine
1-{2-[(3-chloro-2-methylphenyl)carbamoyl]acetyl}piperidine-3-carboxylic acid