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(1R,5R)-N,N-dimethyl-6-[2-(3-methylphenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-{[1-(4-chlorophenyl)ethyl]amino}-N-(2,3-dimethylphenyl)acetamide
dimethyl(2-{2-[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
4-{1-[4-(6-methoxypyridin-2-yl)phenyl]ethyl}morpholine
4-(2-hydroxy-4-methylbenzoyl)piperazine-2-carboxylic acid
[(1-ethylpiperidin-3-yl)methyl](methyl){[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
N-[2-({1,9-dioxaspiro[5.5]undecan-4-yl}amino)ethyl]-4-methoxybenzene-1-sulfonamide
6-{[(3S)-2-oxoazepan-3-yl]amino}-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-(1-phenylcyclopentanecarbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-ethyl-2-[1-ethyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(oxolan-2-ylmethyl)acetamide
N-[(3R,5S)-1-(furan-3-ylmethyl)-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-5-hydroxypyrazine-2-carboxamide
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}({[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl})methylamine
4-{4-[(4-ethylphenyl)methyl]piperazin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-(dimethylamino)-2-(2-methylphenyl)acetamide
7-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-tert-butyl-N-cyclopropyl-4-hydroxypyrimidine-5-carboxamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(2-hydroxy-2-phenylethyl)-N,5-dimethyl-1H-pyrazole-4-carboxamide
4-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-4-oxobutane-1-sulfonamide
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-benzyl-1-cyclopropyl-5-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[(2-chlorophenyl)methyl]-2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]acetamide
1-phenyl-3-(propan-2-yl)-4-(1-propyl-1H-imidazol-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-cyclopentyl-N-(3,3-diphenylpropyl)-6-oxopiperidine-3-carboxamide
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-(1-methyl-1H-indol-3-yl)acetamide
1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(thiophen-2-yl)butan-1-one
3-(methylsulfanyl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
5-methyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]pyrimidin-2-amine
1-(4-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}phenyl)imidazolidin-2-one
1-{[3-(morpholine-4-carbonyl)-1H-pyrazol-5-yl]methyl}-1H-indole
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-{[3-(methylsulfanyl)phenyl]methyl}propanamide
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
5-(oxan-4-yl)-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine
3-(6,8-dimethoxy-4-methylquinolin-2-yl)aniline
{[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(3-methylbutyl)amine
4-{7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}pyridin-2-amine
6-(4-fluorophenyl)-2-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]pyridine-3-carboxylic acid
2-{2-[(dimethylamino)methyl]-4-(pyrimidin-2-yl)phenoxy}-N-{[3-(trifluoromethyl)phenyl]methyl}acetamide
8-[(3-hydroxyphenyl)methyl]-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{1-[2-(3-methoxyphenyl)ethyl]-1H-imidazol-2-yl}-2,4-dimethyl-1,3-thiazole
2-(2-{methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
3-({2-[1-(2,3-dihydro-1-benzofuran-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-1-[4-(1,3-thiazol-2-yl)piperazin-1-yl]ethan-1-one
4-(furan-2-ylmethyl)-3-(3-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]acetamide
6-(benzyloxy)-4-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-1-(2-methylpropyl)-1,4-diazepan-2-one
2-(1-{1-[(2-methyl-1-benzothiophen-3-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
N-ethyl-N,8-dimethyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
2-{[1-(2-methylpyridin-4-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-4-(propan-2-yl)morpholine
N-cyclohexyl-1-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-oxopyrrolidine-3-carboxamide
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-1-ethyl-6-oxopiperidine-3-carboxamide