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(1S,5R)-N-(2H-1,3-benzodioxol-5-yl)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[2-(5-cyano-2-methyl-1H-indol-3-yl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
methyl[(4-methyl-1H-imidazol-5-yl)methyl][3-(oxolan-2-yl)propyl]amine
1-(diethylamino)-3-[2-methoxy-5-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
7-[4-methyl-3-(2-oxoimidazolidin-1-yl)benzoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}ethan-1-one
(3S,4S)-4-methyl-1-{2-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3,4-diol
1-(furan-2-ylmethyl)-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
1-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-4-propyl-1,4-diazepane
1-(2-aminoethyl)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(1,3-dihydroxypropan-2-yl)pyrrolidin-3-yl]-2-methoxy-5-methylbenzamide
2-[(2-hydroxyethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-(4-ethylbenzenesulfonyl)-2,8-diazaspiro[4.5]decane
4-[1-(pyrrolidine-1-sulfonyl)piperidin-3-yl]benzoic acid
1-(2-methoxyphenyl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyridin-4-ylsulfanyl)acetamide
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-(3-chloro-1H-1,2,4-triazol-5-yl)propan-1-one
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-(4-methylphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-phenylpyrrolidin-2-one
N-butyl-4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
5-methoxy-4-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-2-carboxamide
2-{3-[({2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}carbamoyl)amino]phenyl}acetamide
methyl 1-[(3S,5S)-5-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]carbamoyl}-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(1R,5R)-3-methanesulfonyl-6-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-6-(2-methoxyethyl)-3-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[({4-[3-(1H-pyrazol-3-yl)phenyl]phenyl}methyl)amino]propan-1-ol
1-(furan-2-ylmethyl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]piperidine-4-carboxamide
1-[4-(7-{[4-(benzyloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)phenyl]ethan-1-one
7-[2-(thiomorpholin-4-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
(3aR,6aR)-2-cyclohexyl-5-[6-(methoxymethyl)pyrimidin-4-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(1,2-benzoxazol-3-yl)-1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)ethan-1-one
N-benzyl-1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carboxamide
2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]-2-methoxy-6-methylbenzamide
N-[3-(4-{[2-(2-methoxyphenyl)ethyl]amino}piperidin-1-yl)phenyl]pyridine-3-carboxamide
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-[(4-chlorophenyl)methyl]-N-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
2-({spiro[2.5]octan-1-ylmethyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
methyl 2-{3-[({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]-1H-indol-1-yl}acetate
3-benzyl-5-(oxolan-3-yl)-1H-1,2,4-triazole
N-[(1R,3R)-3-aminocyclopentyl]-2,6-dichlorobenzene-1-sulfonamide
(1-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)(pyridin-3-yl)methanol
3-[5-(5-chlorothiophen-2-yl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-(naphthalen-2-yloxy)propanamide
ethyl 4-{[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
4-[(2-aminopyridin-3-yl)methyl]-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
methyl 1-methyl-2-(1,2,3,4-tetrahydroisoquinolin-5-yl)-1H-1,3-benzodiazole-5-carboxylate