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1-cyclohexanecarbonyl-4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazine
{[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]sulfamoyl}diethylamine
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-2-(3-methyl-1H-pyrazol-1-yl)acetamide
1-(5-amino-4-chloro-1H-pyrazole-3-carbonyl)-3-[(dimethylamino)methyl]piperidin-3-ol
3-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]methyl}quinoline
5-methoxy-9-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1-oxa-9-azaspiro[5.5]undecane
4-methyl-2-(1-{2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidin-4-yl)-1H-1,3-benzodiazole
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
4-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)-1H-pyrazole-3-carboxylic acid
2-(4-methoxyphenyl)-5-[(3-propoxypiperidin-1-yl)methyl]pyrimidine
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
7-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2,4-dimethylquinoline
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-{spiro[2.5]octan-1-ylmethyl}propanamide
(2S,4R)-4-(2-cyclopropylacetamido)-N,N-diethyl-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
methyl (2S)-2-{[5-(4-methylpiperidine-1-carbonyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridin-3-yl]formamido}-3-phenylpropanoate
dimethyl[2-(2-{1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-4-yl}-1H-imidazol-1-yl)ethyl]amine
2,3-dimethyl-7-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-{4-[3-({[(2-methylphenyl)methyl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
N-ethyl-N-(oxan-4-ylmethyl)-4-(1H-pyrazol-3-yl)benzamide
6-[(4aS,8aR)-1-(3-methoxypropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]pyridine-2-carbonitrile
3-chloro-N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-4-fluoro-1-benzothiophene-2-carboxamide
N-methyl-1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidine-3-carboxamide
N'-(4-methylphenyl)-N-[2-(2-oxopyrrolidin-1-yl)ethyl]propanediamide
6-ethyl-5-methyl-N4-[2-(1,3-thiazol-2-yl)ethyl]pyrimidine-2,4-diamine
ethyl 2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxylate
2-(5-amino-1,3,4-thiadiazol-2-yl)-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]ethan-1-one
1-(dimethylamino)-2-{4-[(4-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
N-{[(2S,4S)-1-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-4-fluoropyrrolidin-2-yl]methyl}-3-methylbutanamide
2-methyl-4-{5-[({1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}amino)methyl]thiophen-2-yl}but-3-yn-2-ol
2-[(4-fluorophenyl)methyl]-4-(pyridine-3-sulfonyl)morpholine
(2S)-N2-[(4-methoxyphenyl)methyl]-N2-(pyridin-4-ylmethyl)pyrrolidine-1,2-dicarboxamide
N-[(1R,2S)-2-(methoxymethyl)cyclopentyl]-4-sulfamoylbenzamide
methyl 3-[4-(methylsulfanyl)benzoyl]-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-methoxy-6-[3-(1-methyl-1H-pyrazol-3-yl)phenyl]pyrimidine
5-[(4-fluorophenyl)methyl]-3-(oxan-4-yl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
2-(3,5-dichlorophenyl)-5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]pyrimidin-4-ol
5-(phenoxymethyl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1H-pyrazole-3-carboxamide
1-(2-benzylphenyl)-3-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}urea
2-methoxy-3-{4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}pyrazine
1-(carbamoylmethyl)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]piperidine-3-carboxamide
2-amino-4-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1,3-benzothiazole-6-carboxamide
N-[(2-{2-[(dimethylsulfamoyl)amino]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
2-{4-[(2,4-dimethoxyphenyl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
1-(1-benzofuran-2-carbonyl)-4-(cyclopropylmethyl)-1,4-diazepan-5-one
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(3S,4R)-4-(4-fluorophenyl)-1-[3-(2-oxoazepan-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
[3-({1-[5-(methoxymethyl)thiophene-2-carbonyl]pyrrolidin-3-yl}methyl)phenyl]methanol
5-{1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1H-1,2,3-triazol-4-yl}-2-(3-methylphenyl)pyrimidine
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-2,3-dimethylquinoxaline-6-carboxamide
1-(4-fluorophenyl)-4-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl)piperazine