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(2S,4S)-1-[(2-aminopyridin-3-yl)methyl]-N-ethyl-4-[2-(propan-2-yloxy)acetamido]pyrrolidine-2-carboxamide
1-[3-(2-methylphenyl)phenyl]-N-(oxan-3-ylmethyl)piperidin-4-amine
1-[2-(benzyloxy)ethyl]-4-(1H-pyrazole-3-carbonyl)-1,4-diazepan-6-ol
3-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-N-(2-ethoxyphenyl)-3-oxopropanamide
N-(3-cyclopentylpropyl)-N-methyl-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
4-{4-[(4-methylphenyl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-(2-hydroxyethyl)-N-methyl-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
3-chloro-N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}benzamide
N-methyl-4-[2-(methylsulfanyl)ethyl]-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
{2-[2-(2-methoxypyrimidin-5-yl)-1H-imidazol-1-yl]ethyl}dimethylamine
6-[4-(piperidin-1-ylmethyl)benzoyl]-5,6,7,8-tetrahydro-1,6-naphthyridine
4-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-(propan-2-yl)pyrimidine
N-[(4-acetylmorpholin-2-yl)methyl]-5-phenoxyfuran-2-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-2-(morpholin-4-yl)pyrimidine-5-carboxamide
1-[4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
N5-cyclohexyl-1-cyclopropyl-N3-methyl-4-oxo-N3-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
N-(1-ethoxy-2-methylpropan-2-yl)-4-(3-hydroxy-3-methylbutyl)benzamide
8-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 2-{[2-(4-fluorophenyl)ethyl]sulfamoyl}-6-(pent-4-enoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(cyclohex-1-en-1-yl)-5-(methanesulfonylmethyl)pyridine
{1-ethyl-5-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
4-[1-(2H-1,3-benzodioxol-5-yl)-1H-imidazol-2-yl]-1-(2-methoxyethyl)piperidine
N-(oxolan-2-ylmethyl)-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
3-(4-phenylbenzoyl)-1-(1H-pyrazole-4-carbonyl)piperidine
2-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,6-dimethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
1-(cyclohexylmethyl)-5-[4-(2-hydroxyethyl)piperidine-1-carbonyl]piperidin-2-one
N-(3-aminopropyl)-6-(2-fluoro-4-methoxyphenyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-methyl-4-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-2-carbonyl}piperazine
(1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-2-phenylethyl)(methyl)(pyridin-3-ylmethyl)amine
2-[benzyl(methyl)amino]-N-[2-(pyrazin-2-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
(4aS,8aR)-1-(4-hydroxybutyl)-6-(quinolin-4-yl)-decahydro-1,6-naphthyridin-2-one
2-{1-[(1R,2R)-2-(benzyloxy)cyclopentyl]-1H-imidazol-2-yl}pyridine
1-({methyl[1-(1,2-oxazol-3-yl)ethyl]carbamoyl}methyl)piperidine-4-carboxamide
(1S,5R)-6-(2-methoxypyridine-4-carbonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
8-(2-fluorobenzenesulfonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(3R,4R)-4-cyclopropyl-3-methyl-1-(1-phenylpiperidin-4-yl)piperidin-4-ol
3-[3-({[3-(2-amino-1,3-thiazol-4-yl)propyl]amino}methyl)-1H-indol-1-yl]propanamide
4-(hydroxymethyl)-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)benzamide
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(prop-2-en-1-yl)acetamide
1-[(4-fluorophenyl)methyl]-4-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-1,4-diazepane
N-{[1-(propan-2-yl)piperidin-4-yl]methyl}pyrrolidine-1-sulfonamide
dimethyl(1-{3-[2-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]phenyl}ethyl)amine
1-cyclopentyl-4-(2-methylpyrimidin-4-yl)-1,4-diazepane-6-carboxylic acid
1-benzyl-4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-2-one
4-{5-[1-(5-ethyl-1,3-oxazole-4-carbonyl)pyrrolidin-2-yl]thiophene-2-carbonyl}morpholine
methyl 5-cyano-2-methyl-6-[3-(pyridin-3-yl)azetidin-1-yl]pyridine-3-carboxylate
7-(pyrrolidine-1-sulfonyl)-2-{spiro[2.4]heptane-1-carbonyl}-1,2,3,4-tetrahydroisoquinoline
2-amino-6-[4-(1H-imidazol-1-yl)phenyl]-4-(2-methyl-1H-imidazol-4-yl)pyridine-3-carbonitrile