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(3S,4R)-1-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine-4-carbonitrile
N-cyclopentyl-1-[1-(2,5-dimethoxybenzenesulfonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
dimethyl({[4-methyl-5-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
2-(dimethylamino)-N-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}-4-methylpyrimidine-5-carboxamide
4-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-1-oxaspiro[4.5]decan-2-one
2-methyl-5-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
7-(4-chlorophenyl)-2-(pyrimidin-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-1-(6-methylpyridin-3-yl)urea
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-(1H-1,2,4-triazol-1-yl)propan-1-one
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
3-(propan-2-yl)-5-[(2S)-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
N-[3-(1H-imidazol-1-yl)propyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
2-ethyl-5-({4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)pyrimidine
2-{1-[(4-fluorophenyl)methyl]-4-(1-propylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-2-(1H-pyrazol-1-yl)butan-1-one
1-{2-[(3S,4S)-3-(dimethylamino)-4-hydroxypyrrolidin-1-yl]-2-oxoethyl}-3-methyl-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-[1-(cyclohex-3-en-1-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]pyridine
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-{[2-(trifluoromethoxy)phenyl]methyl}urea
1-[(4-fluorophenyl)methyl]-4-(1H-pyrrole-3-carbonyl)-1,4-diazepane
14-[(E)-2-(furan-2-yl)ethenyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
8-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
5-benzyl-4-(3-hydroxypropanoyl)-1-(2-methylphenyl)piperazin-2-one
3-cyclopropyl-3-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(4-sulfamoylphenyl)urea
2-amino-4-(2,5-dimethoxyphenyl)-6-(6-methoxypyridin-3-yl)pyridine-3-carbonitrile
3-butyl-1-methyl-4-(1-methyl-1H-indole-4-carbonyl)piperazin-2-one
2-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)-N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]acetamide
N-ethyl-N-methyl-6-{4-[(1-methyl-1H-indol-2-yl)methyl]piperazin-1-yl}pyrimidin-4-amine
(2R,4S)-4-hydroxy-1-(3-hydroxy-4-methylbenzoyl)piperidine-2-carboxylic acid
8-[(5-methylfuran-2-yl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,4S)-2-methyl-5-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-2,5-diazabicyclo[2.2.1]heptane
3-[4-(pyrimidin-4-yl)piperazin-1-yl]-1,2-benzothiazole
6,7-dimethoxy-2-[1-(oxolane-3-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
1-[2-(1-{4-[(2-hydroxyethyl)sulfanyl]benzoyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
2-amino-N-[3-(cyclopentyloxy)propyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-1,4-diazepan-2-one
N-(3-fluoro-4-methylphenyl)-3-{[1-(4-methanesulfonylphenyl)ethyl]amino}propanamide
2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-(4-methoxy-2-methylphenyl)acetic acid
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1-ethyl-5-methyl-1H-pyrazole-4-carboxamide
N-({1-[(2E)-but-2-en-1-yl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)adamantane-1-carboxamide
4-{3-[(3-hydroxypropyl)carbamoyl]piperidin-1-yl}-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
4-[5-(2-methoxyethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl]benzamide
N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
1-[5-(4-methoxyphenyl)furan-2-carbonyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine
4-{[2-(3,4,5-trimethoxyphenyl)phenyl]methyl}morpholine
2-(2-chloro-4-fluorophenyl)benzamide
4-cyclopentyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrimidin-2-amine
1-{2-[(4-cyclobutyl-6-methylpyrimidin-2-yl)(methyl)amino]ethyl}piperidin-2-one
(2S)-1-{2-[(2-ethoxyphenyl)carbamoyl]acetyl}-N,N-dimethylpyrrolidine-2-carboxamide