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7-cyclopentyl-2-[2-(6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-(2-fluorophenyl)-3-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)propanamide
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]propanamide
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]benzamide
[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl](pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
4-[2-(2,3-dimethylphenoxy)ethyl]-1,2-dihydropyridin-2-one
N'-(3,5-dimethylphenyl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]propanediamide
1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
N-(1-methyl-1H-indazol-3-yl)-2-(4-{1H-pyrazolo[3,4-b]pyridin-4-yl}-1H-pyrazol-1-yl)acetamide
1-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)-1H-1,2,4-triazole
{[5-(4-chloro-2-fluorophenyl)furan-2-yl]methyl}[1-(1H-1,2,4-triazol-5-yl)ethyl]amine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-3-carboxamide
2-(4,5-dichloro-1H-imidazol-1-yl)-N-[1-phenyl-3-(propan-2-yl)-1H-pyrazol-5-yl]acetamide
N-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]pyridine-2-carboxamide
1-(3-chlorophenyl)-4-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-(3-fluorophenyl)propan-1-one
N-cyclopropyl-N-[(7-methoxy-2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}quinolin-3-yl)methyl]-2-(thiophen-3-yl)acetamide
3-methyl-N-(1-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
5-[1-(ethanesulfonyl)ethyl]-1-(3-methylphenyl)-3-phenyl-1H-1,2,4-triazole
4-phenyl-3-({1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2R)-1-(3-methoxy-5-methylthiophene-2-carbonyl)-2-(methoxymethyl)pyrrolidine
methyl 5-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylate
6-cyano-N-[2-(dimethylamino)ethyl]-N-[(3-methylthiophen-2-yl)methyl]pyridine-3-carboxamide
1-cyclopentyl-5-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]piperidin-2-one
(4S)-3-{2-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-oxoethyl}-4-(propan-2-yl)-1,3-oxazolidin-2-one
4-(3-hydroxypropanoyl)-5-methyl-1-(2-phenylphenyl)piperazin-2-one
N-(butan-2-yl)-5-(propan-2-yl)-N-(pyridin-4-ylmethyl)-1,2-oxazole-3-carboxamide
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}({[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl})amine
N-{2-[2-(2,3-difluoro-6-methoxyphenyl)-1H-imidazol-1-yl]ethyl}pyridin-3-amine
2-{5-[2-(methylsulfanyl)ethyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}acetic acid
(2S,4R)-4-(4-{2-[(3-fluoro-4-methylphenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
3-(2,5-dioxoimidazolidin-4-yl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}propanamide
N-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
N-(3-hydroxypropyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-3-carboxamide
2-(3-hydroxyphenyl)-1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
5-(4-acetyl-4-phenylpiperidine-1-carbonyl)-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
N-benzyl-1-{[5-(methoxymethyl)furan-2-yl]methyl}-N-methylpiperidin-3-amine
1-phenyl-4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1,4-diazepane
N-(4-methylphenyl)-5-{[4-(oxolane-2-carbonyl)piperazin-1-yl]methyl}-1,3-thiazol-2-amine
1-[2-(morpholin-4-yl)butanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)methyl]methanesulfonamide
3-{[5-(1-benzofuran-2-yl)-1,2,4-triazin-3-yl](methyl)amino}-1-phenylpropan-1-ol
2,5-dimethyl-N-{[7-(3-phenylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}furan-3-carboxamide
6-phenyl-5-[4-(piperidine-3-carbonyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
3-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-1-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]urea
7-(5-hydroxypyrazine-2-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-methyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1H-indole-6-carboxamide
N-[(4-fluorophenyl)methyl]-3-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]aniline
(4S,6R)-N-(4-butanamido-3-methoxyphenyl)-6-methyl-2-sulfanylidene-1,3-diazinane-4-carboxamide
1-{2-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione