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2-{4-[(3-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}-5,6,7,8-tetrahydroquinoline-3-carbonitrile
(3S,4S)-1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(propan-2-yloxy)pyrrolidin-3-ol
1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
3-(1H-1,2,3-benzotriazol-5-yl)-1-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]urea
3-[1-(cyclopropanesulfonyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
4-(1-benzyl-1H-imidazol-2-yl)-1-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]piperidine
N-{4-[1-(2,6-dimethoxypyridin-3-yl)-1H-imidazol-2-yl]phenyl}acetamide
N,3,4,7-tetramethyl-N-(1-methylpyrrolidin-3-yl)-1H-indole-2-carboxamide
1-{5-[1-(4-cyclohexylpiperazine-1-carbonyl)-6-azaspiro[2.5]octane-6-carbonyl]thiophen-2-yl}ethan-1-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}acetamide
6-tert-butyl-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-{1-oxaspiro[4.4]nonan-3-yl}-1-{2-[2-(pyridin-2-yl)ethoxy]phenyl}urea
3-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-2-ol
N-{[7-fluoro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
2-(4-fluorophenyl)-2-[2-(1-propylpiperidin-4-yl)acetamido]acetic acid
9-[(5-ethylpyridin-2-yl)methyl]-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
N,N-diethyl-3-(5-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)benzamide
[(2-chloro-4-ethoxy-5-methoxyphenyl)methyl](methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
7-{5-methoxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-ethyl-4-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperazine
4-{4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}morpholine
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(1,3-thiazol-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(2-hydroxyethyl)-5-methyl-4-[(oxolan-2-ylmethyl)amino]-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-4-(1H-pyrrole-2-carbonyl)piperazine
6-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-2-carbonitrile
1-benzyl-4-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}pyrrolidin-2-one
6-methyl-2-{[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]methyl}quinolin-4-ol
1-(2-methoxyethyl)-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperazine
methyl 3-[2-(cyclohex-1-en-1-yl)acetyl]-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[1-methyl-5-({4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)-1H-pyrrol-3-yl]ethan-1-one
N-{[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]methyl}-3,5-dimethoxybenzamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
8-(6-methoxyhexanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
5-chloro-3-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-1,2-dihydropyridin-2-one
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylfuran-2-yl)methyl]piperidine
9-{imidazo[1,2-a]pyridin-2-ylmethyl}-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(1R,7S)-3-[(3-methoxyphenyl)methyl]-6-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
(3S,7S)-5-[3-(morpholin-4-yl)propanoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
5-{1-[(2-fluorophenyl)methyl]pyrrolidin-2-yl}-N-(furan-3-ylmethyl)thiophene-2-carboxamide
8-{2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
ethyl 4-(2-methoxyethyl)-1-(3,4,5-trimethoxybenzoyl)piperidine-4-carboxylate
{1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]-3-(3-methylbut-2-en-1-yl)piperidin-3-yl}methanol
2-ethyl-N-methyl-N-(1,2-oxazol-3-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-[2-(4-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
3-chloro-N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-4-fluoro-1-benzothiophene-2-carboxamide
4-(2,4-dioxoimidazolidin-1-yl)-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]benzamide
N3-(1-methoxybutan-2-yl)-N5-[(4-methylphenyl)methyl]-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide