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5-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]oxolane-2-carboxamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
3-(1H-1,2,3,4-tetrazol-1-yl)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-[4-(hydroxymethyl)phenyl]-N-methylpyridine-3-carboxamide
N-(2-methoxyethyl)-1-[1-(pyridine-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)amine
3-[5-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
1-(1-cyclopropylpropan-2-yl)-4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]piperidine
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][3-(methylsulfanyl)propyl]amine
N-{[5-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
(4S)-3,3,4-trimethyl-1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-ol
3-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1-methyl-1H-indole
N-[3-(1H-imidazol-1-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
1-({5-[1-(cyclobutylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-2-(morpholin-3-yl)acetamide
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-N'-(2-methylphenyl)propanediamide
2-methoxy-N-({5-[(2,3,6-trifluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
N-[2-(3-hydroxypiperidin-1-yl)ethyl]-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
2-(2-chlorophenyl)-2-[(1-cyclopropanecarbonylpiperidin-4-yl)formamido]acetic acid
2-(3-{[3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazin-1-yl]methyl}phenoxy)ethan-1-ol
5-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-methyl-3-[methyl(quinolin-2-ylmethyl)amino]butanamide
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[5-(5-fluoro-1H-indole-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
ethyl (1R,5S,6R)-6-[(1,1-dioxo-1λ6-thiomorpholin-4-yl)methyl]-3-azabicyclo[3.1.0]hexane-3-carboxylate
3-{[1-tert-butyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
8-{[4-(trifluoromethyl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]pyrazine-2-carboxamide
2-[(1S,5R)-3-[4-(dimethylamino)benzoyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
3-[4-(3-methoxybenzoyl)piperazin-1-yl]-5-(naphthalen-2-yl)-1,2,4-triazine
N-[3-(furan-2-yl)phenyl]-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-(4-phenylazepan-1-yl)ethan-1-one
N-[1-(4-fluorophenyl)piperidin-4-yl]-4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
{2-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]-1,3-thiazol-4-yl}methanol
methyl 2-(1-{[3-(2-methoxyphenyl)phenyl]carbamoyl}pyrrolidin-3-yl)acetate
6-methyl-2-{[propyl(pyridin-3-ylmethyl)amino]methyl}pyridin-3-ol
[7-(3-methoxy-6-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}benzenesulfonamide
N-{[7-(4-acetylbenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-5-ethyl-1,2-oxazole-3-carboxamide
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,2-dimethylpropanamide
3-hydroxy-N-[(3R,4S)-4-propyl-1-[6-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]propanamide
ethyl 1-{[5-(methoxymethyl)furan-2-yl]methyl}-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
N-(1-cyclopentanecarbonylpiperidin-4-yl)-6-methylimidazo[1,2-a]pyridine-2-carboxamide
N-[1-(ethylcarbamoyl)piperidin-4-yl]-4-hydroxy-2-phenylpyrimidine-5-carboxamide
3-[(3R,4S)-1-(4-chloro-3-fluorobenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
2-[5-(2,7,8-trimethylquinoline-4-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
[(2S,6S)-4-(3-methoxypyrazin-2-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-4H-thieno[3,2-b]pyrrole-5-carboxamide