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2-(propan-2-yl)-6-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
N-butyl-3-[4-(methylamino)pyrimidin-2-yl]benzamide
2-{[4-(1,3-thiazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-3,4-dihydroquinazolin-4-one
1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-[(2-aminopyridin-3-yl)methyl]-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[(3-{[1-(2,4-difluorobenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
2-{4-[(5-chloro-2,3-dimethoxyphenyl)methyl]piperazin-1-yl}pyridine-3-carbonitrile
4-{4-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]piperidin-1-yl}-N-[(2-fluorophenyl)methyl]benzamide
2-(3-chloro-5-methoxybenzoyl)-2,7-diazaspiro[4.5]decan-6-one
N'-(3-ethylphenyl)-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}butanediamide
3-(2-methylphenoxymethyl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine
N-{[(2S,4S)-4-fluoro-1-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}pyrrolidin-2-yl]methyl}pyrrolidine-1-carboxamide
2-[4-({3-[5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
1-cycloheptyl-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(1H-pyrrole-2-carbonyl)piperazine
2-methyl-N-{[4-(morpholin-4-yl)phenyl]methyl}-3-(1H-1,2,4-triazol-1-yl)propanamide
(4aS,7aR)-1-(isoquinoline-3-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{[2-(4-benzylpiperazin-1-yl)ethyl]amino}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[1'-(2-amino-6-methylpyrimidin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
methyl 3-{[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]carbamoyl}propanoate
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-ethyl-1H-indole
N-(1-{7-[(4-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
8-methyl-2-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
2-(1-methylpyrrolidin-3-yl)-9-(2-phenylacetyl)-2,9-diazaspiro[5.5]undecan-3-one
1-({2-[(3-fluorophenyl)methoxy]-3-methoxyphenyl}methyl)azepan-4-ol
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-3-(furan-3-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-hydroxy-1-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
N-(1,2-oxazol-5-ylmethyl)-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1'-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
methyl 5-{[(2,3-dimethoxyphenyl)methyl]amino}-1-ethyl-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(cyclohexylmethyl)-3-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}-3-hydroxypiperidin-2-one
3-methoxy-2-{[(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}phenol
2-(6-methoxynaphthalen-2-yl)-4-[3-(4-methyl-1H-pyrazol-1-yl)propyl]morpholine
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(pyrazin-2-yl)ethyl]benzamide
1-{imidazo[1,2-b]pyridazin-6-yl}-4-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperazine
2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-1-[(3-methylthiophen-2-yl)sulfonyl]piperidine
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
4-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]-5-tert-butylfuran-2-carboxamide
6-[4-(1-methoxyethyl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[(2-chlorophenyl)methyl]-2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-(2-methoxyethyl)acetamide
1-(3-fluoro-5-methylphenyl)-3-[4-(pyrrolidin-1-yl)butyl]urea
1-[5-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-(piperidin-1-yl)propan-2-ol
(2R,3R,6R)-5-(4-methyl-1H-imidazole-5-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(2-methoxyethyl)-3-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)propanamide
1-[(2S)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]-3-(pyridin-4-yl)propan-1-one
5-[(3aS,6aR)-3-[(2-methoxyphenyl)methyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carbonyl]-1,2-dihydropyridin-2-one
N-[4-(3-fluorophenyl)phenyl]-1-[(2-methylpyrimidin-5-yl)methyl]pyrrolidine-2-carboxamide
ethyl 4-[2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamido]piperidine-1-carboxylate
[9-methyl-3-(1,3-thiazole-5-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
4'-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one