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N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-fluoropyridine-4-carboxamide
1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(methylsulfanyl)ethan-1-one
2-(2,3-difluorophenoxymethyl)-N-(oxan-2-ylmethyl)-1,3-oxazole-4-carboxamide
2-(2,3-difluorophenyl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
N-cyclopentyl-3-[(3S,4R)-1-(2-methylpropyl)-4-(morpholin-4-yl)piperidin-3-yl]propanamide
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)(pyridin-3-ylmethyl)amine
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)acetamide
3-[(1-cyclohexylpyrrolidin-3-yl)methyl]-1-(4-sulfamoylphenyl)urea
1-{4-[(2-methoxyphenyl)methyl]piperazin-1-yl}-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-(naphthalen-1-ylmethyl)piperidine-3,5-dicarboxamide
1-cyclobutanecarbonyl-N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]piperidine-4-carboxamide
(4aS,8aR)-1-(3-methoxypropyl)-6-[2-(pyridin-3-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
8-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
[(3R,4R)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
4-{[(2-fluorophenyl)methyl]amino}-1-(2-phenylethyl)pyrrolidin-2-one
N-ethyl-3-(1,2-oxazolidin-2-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
(3S,4R)-1-[(2H-1,3-benzodioxol-5-yl)carbamoyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
(4aS,7aR)-1-[(2E)-hex-2-en-1-yl]-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-ethyl-4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
1-[2-({[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]piperidin-4-ol
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]imidazo[1,2-a]pyridine-6-carboxamide
8-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(2-methyl-1,3-thiazole-4-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
4-(2,6-dimethoxy-4-methylphenyl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine
N-{[(2S)-1-ethylpyrrolidin-2-yl]methyl}-2-(4-methyl-1,4-diazepan-1-yl)acetamide
methyl (2R,4S)-1-(dimethylsulfamoyl)-4-hydroxypiperidine-2-carboxylate
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-(piperidin-1-ylmethyl)piperidin-2-one
2-cyclopropyl-N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
5-ethyl-2-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}pyrimidine
methyl 2-hydroxy-5-{[(1-methylpiperidin-4-yl)(pyridin-3-ylmethyl)amino]methyl}benzoate
methyl 3-[4-(furan-2-carbonyl)-6-[(3-methoxyphenyl)methoxy]-2-oxo-1,4-diazepan-1-yl]propanoate
5-({4-[(2-fluorophenyl)methyl]piperidin-1-yl}methyl)-2-methylpyridine
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-6-ethyl-2-methylpyrimidin-4-amine
4-(2,6-dimethylpyridin-3-yl)-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}pyrimidin-2-amine
3-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1-(difluoromethyl)-1H-pyrazole
4-[4-oxo-7-(5-propylpyrimidin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
1-methyl-3-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}-1H-indole
N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
2-[(3-{[2-(pyridin-4-yl)ethyl]carbamoyl}phenyl)amino]acetic acid
1-methyl-4-[1-(2-methylpropyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-3-phenyl-1H-pyrazole
5-(azepane-1-carbonyl)-N-(1-benzylpiperidin-4-yl)-1-(butan-2-yl)-4-oxo-1,4-dihydropyridine-3-carboxamide
4-{2-ethyl-3H-imidazo[4,5-b]pyridin-6-yl}-3,5-dimethyl-1H-pyrazole
(2R)-N-[2-(naphthalen-1-yl)propan-2-yl]oxolane-2-carboxamide
N-[2-(3-acetamidophenyl)pyridin-3-yl]-2-methylpropanamide
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-3-methyl-N-[(3S)-2-oxoazepan-3-yl]thiophene-2-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
2-chloro-N-(2-{imidazo[1,2-a]pyridin-6-ylformamido}ethyl)benzamide