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N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-1,4-dithiepan-6-amine
4-(4-phenyl-1,4-diazepane-1-carbonyl)-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(pyrazin-2-yl)ethan-1-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-methyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
3-(1-butyl-3-methyl-1H-pyrazol-5-yl)-1-[1-(4-methanesulfonylphenyl)ethyl]urea
1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
(2S,4R)-4-amino-1-[3-(3-hydroxyquinoxalin-2-yl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]-1,3-benzoxazole
2-{1-[(2-methylphenyl)methyl]-4-{[3-(methylsulfanyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
4-(1-benzoylpiperidin-3-yl)-5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidine
1-[4-(azocane-1-carbonyl)phenyl]imidazolidine-2,4-dione
6-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]pyridine-3-carboxylic acid
methyl 2-[1-(1-cycloheptyl-6-oxopiperidin-3-yl)-N-methylformamido]acetate
4-{1-[1-(pyridin-2-yl)piperidine-3-carbonyl]piperidin-4-yl}thiomorpholine
8-cyclopropanecarbonyl-2-(dimethyl-1,3-oxazole-4-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-cyclopentyl-1-[(4-methoxyphenyl)methyl]-5-(pyridine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(1-carbamoylcyclopentyl)-4-(piperidin-1-ylmethyl)benzamide
4-{4-[(3,5-dimethoxyphenyl)methyl]piperazin-1-yl}-2-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-(1H-indol-3-yl)-1-(4-{2-[2-(4-methoxyphenyl)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)ethan-1-one
5-[5-(morpholin-4-ylmethyl)pyridin-2-yl]isoquinoline
7-cyclopentyl-2-{[6-(dimethylamino)pyridin-3-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-2-[4-(hydroxymethyl)phenyl]ethan-1-one
3-(5-methylthiophen-2-yl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1H-pyrazole-5-carboxamide
4-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}-1-[4-(propan-2-yl)phenyl]pyrrolidin-2-one
2-(2-cyclopentylacetyl)-N-(2-methoxyethyl)-1,2,3,4-tetrahydroisoquinoline-8-sulfonamide
4-{1-[3-(morpholin-4-yl)propyl]-4-phenyl-1H-imidazol-5-yl}phenol
5-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-2-methylphenol
N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]quinoline-2-carboxamide
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
1-cyclopentanecarbonyl-N-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-amine
2-amino-7-[5-(oxolan-2-yl)thiophene-2-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{4-[2-(1-ethyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]phenyl}-5-methylpyrrolidin-2-one
5-{[6-hydroxy-4-(1H-imidazol-2-ylmethyl)-1,4-diazepan-1-yl]methyl}-N,N-dimethylfuran-2-carboxamide
2-[(cyclopropylmethyl)sulfanyl]-1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-{2-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-oxazol-3-ol
3-{[ethyl(methyl)amino]methyl}-1-[(2-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
(1R,2R,6S,7S)-4-{5-[1-(piperidin-1-yl)ethyl]furan-2-carbonyl}-4-azatricyclo[5.2.1.02,6]decane
methyl 3-[2-(3-fluorophenyl)acetyl]-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1R,5R)-3-cyclobutanecarbonyl-6-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-(2-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperidin-3-yl}ethyl)methanesulfonamide
N-({1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidin-3-yl}methyl)-2,3-dihydro-1-benzofuran-7-carboxamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(2,6-dimethylpyrimidine-4-carbonyl)piperidine-3-carboxylate
N-(2-hydroxyethyl)-1-{1-[(2-methoxynaphthalen-1-yl)methyl]piperidin-3-yl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-[1-(3-methylbutyl)-4-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-yl]ethan-1-ol
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-acetamido-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)benzamide
4-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3-phenyl-1H-pyrazole
1-[(4-methanesulfonylphenyl)methyl]-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazine
2-[(4aR,7aS)-4-[(3,5-dimethylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide