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N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(1H-imidazol-1-yl)propanamide
2-(thiomorpholine-4-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
N-cyclopentyl-2-[(2-methylpropyl)(pyridin-2-ylmethyl)amino]propanamide
3-{2-[5-(4-acetylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,3-oxazinan-2-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylspiro[2.4]heptane-1-carboxamide
(1S,5R)-3-[2-(2-chloro-6-fluorophenyl)acetyl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S,4S)-N-ethyl-1-(2-hydroxyethyl)-4-(4,5,6,7-tetrahydro-1-benzothiophene-2-amido)pyrrolidine-2-carboxamide
methyl 3-(2-chlorobenzenesulfonamido)-5-({[5-(methoxymethyl)furan-2-yl]formamido}methyl)benzoate
7-methoxy-3-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
(3S)-2-(1H-1,2,3-benzotriazole-5-carbonyl)-N-tert-butyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-[2-(dimethylamino)ethyl]-5-oxo-N-[2-(1,3-thiazol-4-yl)ethyl]pyrrolidine-3-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-4-(thian-4-yl)piperazine
(2E)-N-({5-fluoro-7-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
3-{1-[4-(1H-imidazol-1-yl)butanoyl]piperidin-3-yl}benzoic acid
(4aS,8aR)-6-[(5-ethylpyridin-2-yl)methyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
ethyl 4-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
methyl (1R,3S,3aR,6aS)-3-(2-chloro-6-fluorophenyl)-1-ethyl-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
(2S,4R)-4-[(adamantan-2-yl)amino]-N-(propan-2-yl)-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(oxan-4-yl)ethyl]acetamide
3-(1-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1-(pyrrolidin-1-yl)propan-1-one
1-cyclohexyl-4-(pyrazine-2-carbonyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
N-[1-(cyclohex-1-en-1-yl)ethyl]-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(4-ethylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-cyclohexyl-3-(cyclopropylmethyl)-N-ethyl-N-(2-hydroxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}propanamide
N-(2-chlorophenyl)-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
[1-(5-{[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-yl]methanol
(1S,5R)-6-(cyclopropylmethyl)-3-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
5-(methoxymethyl)-N-[4-(5-methyl-4-{[2-(phenylsulfanyl)acetamido]methyl}-1,3-oxazol-2-yl)phenyl]furan-2-carboxamide
methyl 2-(2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamido)acetate
methyl 1-(naphthalen-2-ylmethoxy)-2-oxo-8-(quinolin-6-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
N-[2-(4-fluorobenzenesulfonyl)ethyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-methyl-5-(pyrrolidin-2-yl)-N-(quinolin-5-ylmethyl)thiophene-2-carboxamide
[(5-chlorofuran-2-yl)methyl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
2-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyridine-4-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-3-methylbut-2-enamide
(3S,9aR)-3-(4-aminobutyl)-8-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(2-{4-[1-(dimethylamino)ethyl]phenyl}-1H-imidazol-1-yl)propan-1-ol
N-[(3-chlorophenyl)methyl]-3-(methylsulfanyl)-N-propylpropanamide
2-{4-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
1-(4-ethylpiperazin-1-yl)-3-{3-[({[3-(methylsulfanyl)phenyl]methyl}amino)methyl]phenoxy}propan-2-ol
2-[4-(1H-1,3-benzodiazol-2-ylmethyl)-1-[(4-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
1-cyclopropanecarbonyl-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]piperidine-4-carboxamide
2-(3-phenylpropyl)-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
1-{1-benzyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}cyclopropane-1-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}acetamide