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N-(5-methyl-1,2-oxazol-3-yl)-2-(oxane-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
9-methoxy-N-[(2-methoxyphenyl)methyl]-3-[(6-methylpyridin-2-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-ethyl-4-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
(1-{[(7-methoxy-4-methylquinazolin-2-yl)(methyl)amino]methyl}cyclopentyl)methanol
3-methyl-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]but-2-en-1-one
4-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}pyridin-2-amine
4-{2-[bis(propan-2-yl)carbamoyl]-3-methoxyphenyl}thiophene-2-carboxamide
2-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}-4-(pyridin-2-yl)phenol
[3-(3-methoxypropyl)-1-(2,3,6-trifluorobenzoyl)piperidin-3-yl]methanol
1-{2-[2-(3-methoxyphenyl)acetamido]ethyl}-N-[(4-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
(3R,4R)-4-(hydroxymethyl)-1-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]piperidin-3-ol
methyl (2S)-1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxylate
N-[(3R,4S)-4-(4-methoxyphenyl)-1-methylpyrrolidin-3-yl]piperidine-1-sulfonamide
3-[1-(1-benzothiophen-2-ylmethyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
N-[2-(2-methyl-1H-indol-1-yl)ethyl]-2-(1-methyl-3-oxopiperazin-2-yl)acetamide
2-methoxy-4-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridine-3-carbonitrile
1-{1-[1-(5-chloro-2-fluorobenzoyl)piperidin-4-yl]ethyl}-4-methylpiperazine
2-(2,6-dimethoxyphenyl)-2-{[(5-ethylpyridin-2-yl)methyl](methyl)amino}acetic acid
2-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-(oxan-4-yl)-5-{1H,4H,6H,7H-pyrano[4,3-c]pyrazol-3-yl}-1H-1,2,4-triazole
methyl (2S,4S)-1-methyl-4-[2-(3-methyl-1,2-oxazol-5-yl)acetamido]pyrrolidine-2-carboxylate
7-(1H-indole-6-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-6-methyl-3-[4-(4-methylphenyl)piperazine-1-carbonyl]-2-propyl-1,4-dihydropyridin-4-one
6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-(pyridine-2-carbonyl)-1,4-diazepan-2-one
3-{3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidine-1-carbonyl}pyridin-1-ium-1-olate
[(2-butyl-1H-imidazol-4-yl)methyl]({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)methylamine
4-(4-{[(5-methyl-1H-pyrazol-3-yl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
4-(2,5-dimethylthiophen-3-yl)-2-{4-[4-(2-methoxyethyl)piperazine-1-carbonyl]-5-methyl-1H-pyrazol-1-yl}pyrimidine
4-methoxy-2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
5-{3-[4-(5-amino-3-methyl-1H-pyrazol-1-yl)phenyl]-1,2,4-oxadiazol-5-yl}-1-ethylpiperidin-2-one
2-(2-chloro-4-{[cyclopropyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)propanoic acid
5-acetyl-N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)thiophene-3-carboxamide
N-(furan-2-ylmethyl)-4-methoxy-N-(3-methylbutan-2-yl)cyclohexane-1-carboxamide
2-(phenylamino)-N-(2,2,2-trifluoroethyl)pyrimidine-5-carboxamide
2-(2,4-dichlorophenoxy)-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]acetamide
N-[3-(pyridin-2-yl)propyl]-6-(pyridin-3-yl)pyridine-3-carboxamide
ethyl 1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
[(4aS,8aR)-6-(6-chloro-2-methylquinoline-4-carbonyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
N-{[3-(quinolin-8-yl)phenyl]methyl}cyclopropanamine
{[(3S,4R)-1-(5-fluoropyrimidin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-{4-phenyl-1-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-1H-imidazol-5-yl}-1-(propan-2-yl)piperidine
dimethyl({2-[(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amino]ethyl})amine
1-(5-ethyl-1,3,4-oxadiazol-2-yl)-4-(3-methoxypropyl)piperazine
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]acetamide
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[3-(pyridin-4-yl)propyl]-1H-pyrazole-4-carboxamide
3-hydroxy-1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
(2S)-2-({2-cyclopentyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)-4-(methylsulfanyl)butan-1-ol
(3-{5-[(2E)-but-2-en-1-yl]-1,2,4-oxadiazol-3-yl}phenyl)methanol
3-[1-(6-aminopyrimidin-4-yl)piperidin-4-yl]-4-benzyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one