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N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-{[(1s,4s)-4-aminocyclohexyl]amino}pyridine-3-carboxamide
methyl 5-cyano-6-[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-2-methylpyridine-3-carboxylate
N-[3-(tert-butylcarbamoyl)-2-methylphenyl]-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
3-(3-{3-[4-(dimethylamino)-5-methylpyrimidin-2-yl]phenyl}-1H-pyrazol-1-yl)propan-1-ol
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]pyrrolidine-2-carboxylate
N,3-dicyclopropyl-N-(3-phenylprop-2-yn-1-yl)-1H-pyrazole-5-carboxamide
6-[4-(ethylsulfanyl)phenyl]-9H-purin-2-amine
2-(4-chloro-2-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}phenoxy)acetic acid
5-ethyl-2,3-dimethyl-N-(3,3,3-trifluoropropyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}propanamide
2-[(3,5-difluorophenyl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
1-[4-(furan-2-yl)benzoyl]-4-(2-methylpropyl)-1,4-diazepan-5-one
(1S,5R)-N-(4-acetylphenyl)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-{1-[(2-methoxyphenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-(propan-2-yl)-1H-pyrazole
4-{5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(1H-imidazol-5-yl)ethyl]-1H-1,2,4-triazol-3-yl}pyridine
methyl[(3-methylpyridin-2-yl)methyl]{[5-(oxan-2-yl)thiophen-2-yl]methyl}amine
3-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)formamido]-3-phenylpropanoic acid
2-{4-[3-(pyridin-3-yl)-1H-pyrazol-1-yl]phenoxy}ethan-1-ol
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amine
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
6-{1-[3-(dimethylamino)benzoyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
ethyl 5-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}benzenesulfonyl)pyrrolidine
9-(3-hydroxypyridine-2-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
2-{5-[2-(dimethylamino)phenyl]-1-(2-hydroxyethyl)-1H-1,2,4-triazol-3-yl}acetamide
N-[(1-hydroxycyclohexyl)methyl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrimidin-2-amine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,4-dimethyl-1,3-oxazole-5-carboxamide
(2R,3S,6R)-5-(1,2-oxazole-3-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[4-(2,5-dimethoxybenzoyl)benzoyl]-N-phenylpiperidin-3-amine
1-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}-2-(4-fluorophenyl)piperidine
4-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-6-fluoro-2-(pyrimidin-5-yl)quinoline
1-(cyclohex-1-en-1-ylmethyl)-3-[5-(5-ethyl-1,3,4-oxadiazol-2-yl)-2-methoxyphenyl]urea
5-[1-(4-chlorobenzenesulfonyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
1-[(2E)-3-phenylprop-2-en-1-yl]-4-{[4-(pyrrolidine-1-carbonyl)-1,3-oxazol-2-yl]methyl}piperazine
2-(2-methyl-1H-indol-3-yl)-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
6-ethyl-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2-methylquinoline-4-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[1-(oxan-4-yl)piperidin-4-yl]benzamide
(1S,5R)-6-(1-methyl-1H-pyrrole-2-carbonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-[(3-fluorophenyl)methyl]piperazine
(2S,4S)-4-amino-1-methyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrrolidine-2-carboxamide
1-(1H-imidazol-1-ylmethyl)-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]cyclopropane-1-carboxamide
4-chloro-1-methyl-3-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-1H-indazole
N-(carbamoylmethyl)-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-[(6-methylpyridin-2-yl)methyl]-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
3-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-(4-sulfamoylphenyl)urea
methyl 1-[(3S,5S)-5-(cycloheptylcarbamoyl)-1-[(4-fluorophenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-6-methoxy-1-methyl-1H-indole-2-carboxamide
9-(1-acetylpiperidine-3-carbonyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-{[2-(diethylamino)pyridin-3-yl]methyl}-1,3-benzothiazole-5-carboxamide