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1-{2-[1-(2-ethylpyrimidine-5-carbonyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
[(2S,6S)-4-(pyridine-4-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
2-[4-(4-cyclopentylpyrimidin-2-yl)piperazin-1-yl]-N-ethylacetamide
3-chloro-N-(2-methoxyethyl)-4-({1-[(4-methylphenyl)methyl]piperidin-4-yl}oxy)benzamide
5-(3-fluorophenoxymethyl)-N-(2-hydroxyethyl)-N-methyl-1H-pyrazole-3-carboxamide
N-[1-(1H-indol-2-yl)ethyl]-N-methyl-4-(4H-1,2,4-triazol-4-yl)benzamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]pyrrolidine-3-carboxylic acid
1-{[1-(4-ethylbenzenesulfonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
N-cyclopropyl-3-{5-[2-(dimethylamino)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-(furan-2-ylmethyl)-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]piperidine-4-carboxamide
N-(1,4-dioxan-2-ylmethyl)-N,15-dimethyl-9-(5-methylthiophen-2-yl)-13-oxo-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
6-amino-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)pyridine-2-carboxamide
1-{[3-chloro-5-methoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}-N-ethylpyrrolidine-3-carboxamide
N-[4-(2-methoxypyridin-3-yl)-2-methylphenyl]pyridine-3-carboxamide
4-methyl-N-(2-{7-[(3,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
2-[3-(3-chlorophenoxymethyl)-5-cyclobutyl-1H-1,2,4-triazol-1-yl]acetic acid
N-(2-{4-[(4-phenylpiperazin-1-yl)methyl]phenoxy}propyl)propanamide
4-(1H-imidazol-1-yl)-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]benzamide
N-(3-methyl-1-propyl-1H-pyrazol-5-yl)-4-(pyrimidin-2-yl)-1,4-diazepane-1-carboxamide
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
1-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]-2-(1-propylpiperidin-4-yl)ethan-1-one
2-[({1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperidin-3-yl}oxy)methyl]pyridine
(2S,4R)-4-amino-N-methyl-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]pyrrolidine-2-carboxamide
N-[1-(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]-2,5-dimethoxybenzamide
2-[2-(2-methylpropoxy)phenyl]-3-(pyrrolidine-1-carbonyl)pyridine
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]oxane-4-carboxamide
(5S)-5-[({[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]pyrrolidin-2-one
4-(2-hydroxypropyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-oxazole-3-carboxamide
2,3-dimethoxy-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(2-methoxyphenoxy)piperidin-1-yl]ethan-1-one
N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4-oxo-3,4-dihydrophthalazine-1-carboxamide
5-fluoro-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-(pyrrolidin-1-yl)pyrimidin-2-amine
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methylacetamide
(3S,4S)-4-(naphthalen-2-yl)-1-(pyridine-2-carbonyl)piperidin-3-ol
2-[(2R,3R)-2-hydroxy-3-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-N-(2-methylbutan-2-yl)acetamide
3-[({1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}oxy)methyl]pyridine
2-cyano-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
2-({[2-(diethylamino)pyridin-3-yl]methyl}amino)pyridine-3-carboxamide
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(1H-1,2,4-triazol-1-yl)propanamide
3-[1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methoxypyridine
3-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1-[1-(pyrazin-2-yl)propan-2-yl]urea
5-[2-(4,5-dimethyl-1H-pyrazol-3-yl)ethyl]-3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazole
1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}(4,4,4-trifluorobutan-2-yl)amine
1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-1,4-diazepan-5-one
N-{1-[3-(pyrrolidin-3-yl)benzoyl]piperidin-4-yl}methanesulfonamide
(3S,4S)-1-[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
methyl 4-{4-[2-(4-chloro-1H-pyrazol-1-yl)acetyl]piperazin-1-yl}benzoate