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N-[1-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]oxolane-3-carboxamide
5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[2-(naphthalen-1-yl)ethyl]-1,2-oxazole-3-carboxamide
3-({[(2-aminopyridin-3-yl)methyl]amino}methyl)-3-hydroxy-1-[(3-methoxyphenyl)methyl]piperidin-2-one
5-{[4-(1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}pentan-1-ol
1-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}-2-(pyrrolidin-1-yl)ethan-1-one
2-(4-ethyl-1,3-thiazol-2-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
[(3R,4R)-1-[(2-chloro-4,5-dimethoxyphenyl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
(3R,4S)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(3-methoxyphenyl)pyrrolidin-3-amine
2-(hydroxymethyl)-2-[(2-methyl-5-propylpyrimidin-4-yl)amino]propane-1,3-diol
N-methyl-N-(1-{1-[2-(4-methylphenoxy)acetyl]piperidin-4-yl}-2-phenylethyl)thiophene-2-carboxamide
N-[(1S,3S)-3-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}cyclopentyl]pyridazine-3-carboxamide
1-{1-[6-(2-methoxyphenyl)pyridazin-3-yl]piperidin-4-yl}propan-1-ol
1-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]-2-(2-phenylethyl)piperidine
(2S)-N-[3-(3-methylphenyl)phenyl]-1-(morpholine-4-carbonyl)pyrrolidine-2-carboxamide
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-(pyridin-3-ylmethyl)piperidin-3-amine
N,N-dimethyl-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
8-[2-(ethylsulfanyl)pyrimidin-5-yl]-2-(morpholin-4-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
2-[3-methyl-4-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-1H-pyrazol-1-yl]ethan-1-ol
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(N-methylmethanesulfonamido)ethyl]acetamide
N-(1,2-oxazol-3-ylmethyl)-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
4-(1H-imidazol-2-yl)-1-[4-(1-phenyl-1H-imidazol-4-yl)benzoyl]piperidine
2-{[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-5-methoxypyridin-4-ol
1-(3-chlorophenyl)-4-[2-hydroxy-4-(methylsulfanyl)butanoyl]piperazin-2-one
2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-4-(thiomorpholine-4-carbonyl)-2,3-dihydro-1H-isoindol-1-one
1-(4-fluorophenyl)-4-[(4-methoxy-3-{2-[1-(pyridine-3-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl]piperazine
3-(2-chlorophenyl)-1-cyclopentyl-3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]pyrrolidine-2,5-dione
3-methyl-2-{2-[2-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl}pyridine
3-({[(5-chlorothiophen-2-yl)methyl]amino}methyl)-1-(cyclopropylmethyl)-3-hydroxypiperidin-2-one
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][(2-fluoro-4,5-dimethoxyphenyl)methyl]methylamine
2-(4-chlorophenyl)-4-(3-methyl-1H-pyrazole-5-carbonyl)morpholine
2-(3-fluorophenoxymethyl)-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]-1,3-oxazole-4-carboxamide
N-[(2-fluorophenyl)methyl]-1-methyl-5-{methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(2,3-dihydro-1H-inden-1-yl)acetamide
2-{[1-(5-methoxypyridin-3-yl)-4-methyl-1H-1,3-benzodiazol-2-yl]methoxy}acetic acid
2-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-4-phenyl-1,2-dihydrophthalazin-1-one
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-1H-1,2,4-triazole-5-carboxamide
6-butyl-2-(4-{[(2-methoxyethyl)(methyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
(2S,4S,5R)-4-[(2,2-difluoroethyl)carbamoyl]-1-methyl-2-(2-methylpropyl)-5-(pyridin-3-yl)pyrrolidine-2-carboxylic acid
1-{2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
2-(3-{1-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
3-[3-({[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]amino}methyl)-1H-indol-1-yl]propanamide
(2E)-1-[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]-3-(pyridin-4-yl)prop-2-en-1-one
6-(azepan-1-yl)-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
4-(dimethyl-1,3-thiazole-5-carbonyl)morpholine-2-carboxylic acid
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
ethyl 3-[(3-methoxyphenyl)methyl]-1-(3-methylthiophene-2-carbonyl)piperidine-3-carboxylate
3-[3-ethyl-4-(4-fluorophenyl)-1-methyl-1H-pyrazol-5-yl]-1-methyl-1-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]urea
6-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one