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2-{4-[2-(methylsulfanyl)pyridine-3-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-4-(1H-pyrazol-1-yl)butan-2-ol
4-(3-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}phenyl)-2-methylbutan-2-ol
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-hydroxy-2-methylpyrimidine-5-carboxamide
4-({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)butan-1-ol
(3aS,6aS)-2-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-(2-aminopyrimidin-4-yl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{2-hydroxy-3-[2-methoxy-4-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
5-{5-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
2-methyl-8-[2-(5-phenyl-4H-1,2,4-triazol-3-yl)ethyl]-2,8-diazaspiro[5.5]undecane
9-[2-(2,3-dimethylphenoxy)ethyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
1-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3-(prop-2-en-1-yl)urea
[3-(2,4-dimethoxypyrimidin-5-yl)phenyl]methanol
1-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-3-[3-(2-oxopyrrolidin-1-yl)propyl]urea
1-[(2-fluorophenyl)methyl]-N-methyl-N-(quinolin-2-ylmethyl)piperidin-3-amine
1-[(5-ethylfuran-2-yl)methyl]-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
5-(4-fluorophenyl)-N-[3-(pyridin-4-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
(2R,3R)-3-amino-1'-(4-hydroxy-3-methoxybenzoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-[(3,4,5-trimethoxyphenyl)methyl]propanamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-ethyl-N,4-dimethyl-1,3-oxazole-5-carboxamide
2,2-dimethylpropyl 3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxylate
N-({1-[(2,3-difluoro-4-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-2-methyl-2-(methylamino)propanamide
1-[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidin-1-yl]but-3-en-1-one
(3S)-4-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-1-ethyl-3-methylpiperazin-2-one
1-(carbamoylmethyl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]piperidine-3-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-1-[3-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]propan-1-one
dimethyl(1-{4-[1-(5-methylpyridin-3-yl)-1H-imidazol-2-yl]phenyl}ethyl)amine
1-(oxane-4-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
(2S,4R)-4-amino-1-(4-cyanobenzenesulfonyl)-N,N-diethylpyrrolidine-2-carboxamide
N-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
1-(azepan-2-ylmethyl)-3-(4-methoxy-2-methylphenyl)urea
2-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-benzofuran-7-carboxamide
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-3-(1H-pyrazol-1-yl)benzamide
1-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]-2-(3-hydroxyphenyl)ethan-1-one
4-(6-aminopyridine-3-carbonyl)-7-(3-chlorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N,2-dimethyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
(1S,4S)-2-(3-chloro-4-methoxyphenyl)-5-(quinolin-6-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
(1R,3S)-3-methoxy-7-[(8-methoxy-2H-chromen-3-yl)methyl]-7-azaspiro[3.5]nonan-1-ol
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}[(2-phenyl-1,3-thiazol-4-yl)methyl]amine
(3aR,6aR)-2-methanesulfonyl-5-[2-(2-methoxyphenyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-[(3-hydroxy-4-methoxyphenyl)methyl]-6-(4-methoxyphenyl)-6,9-diazaspiro[4.5]decan-7-one
N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(3-chloro-4-hydroxyphenyl)acetamide
[1-({[(4-fluoro-3-methoxyphenyl)methyl](methyl)amino}methyl)cyclopentyl]methanol
N,N,6-trimethyl-2-[2-(pyridin-3-yl)pyrimidin-5-yl]quinoline-4-carboxamide
2-(4-{[4-(ethylamino)pyrimidin-2-yl]amino}piperidin-1-yl)acetamide
2,3-dimethyl-7-[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-N-(1,3,4-thiadiazol-2-yl)propanamide
4-(2-{1-[2-(methylamino)pyridine-4-carbonyl]piperidin-2-yl}ethyl)phenol
(3R,5S)-N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide