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1-{3-[(2-methylprop-2-en-1-yl)oxy]phenyl}-5-oxopyrrolidine-3-carboxylic acid
N-[1-(5-methoxy-3-methyl-1H-indole-2-carbonyl)piperidin-4-yl]pyrimidin-2-amine
[(1-methyl-1H-imidazol-2-yl)methyl]({6-methyl-2-[(2-methylphenyl)methoxy]quinolin-3-yl}methyl)amine
(3S,9aR)-3-(4-aminobutyl)-8-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-[5-(1H-imidazol-1-ylmethyl)furan-2-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-(2-methoxyphenyl)-1-(3-methoxypropyl)-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
methyl 9-(oxan-2-ylmethoxy)-7-oxo-3-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[3-(1H-imidazol-1-yl)propyl]-2-(morpholin-3-yl)acetamide
1-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-2-(5-methylfuran-2-yl)-1H-imidazole
4-{4-[3-(hydroxymethyl)morpholine-4-carbonyl]phenyl}-2-methylbutan-2-ol
(3R,4S)-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3,4-dimethylpiperidin-4-ol
(4-{[2-(2-phenylethoxy)phenyl]methyl}morpholin-3-yl)methanol
N,N-diethyl-2-(4-{2-[2-(3-hydroxyphenyl)ethyl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)acetamide
N-(1H-indol-5-ylmethyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-(4-chloro-2-methylbenzoyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-{4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
(benzylsulfamoyl)(methyl)[2-(2-methylpiperidin-1-yl)ethyl]amine
3-[(3R,4S)-4-(morpholin-4-yl)-1-[6-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]propan-1-ol
3-[1-(3-cyclopentylpropyl)piperidin-4-yl]-N-(2-methoxyethyl)propanamide
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-5-oxopyrrolidine-3-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
N,N-dimethyl-3-[(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)methyl]-1,2,4-oxadiazole-5-carboxamide
methyl N-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]carbamate
6-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-amine
2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]-8-fluoroquinoline
(2E)-1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-phenylprop-2-en-1-one
3-(1-methyl-1H-pyrrol-2-yl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1H-pyrazole-5-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[3-(3-methoxypropyl)piperidin-1-yl]ethan-1-one
N-(3-hydroxypropyl)-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-methyl-1H-indole-2-carboxamide
5-{2-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-2-ethyl-6-methyl-3,4-dihydropyrimidin-4-one
(3R,4R)-3-[4-(1,3-benzoxazol-2-yl)piperazine-1-carbonyl]-1-methylpiperidin-4-ol
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-4-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]butanamide
2-{[6-(pyrrolidin-1-yl)pyridazin-3-yl]oxy}-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
2-[3-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-3-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[(2-methylprop-2-en-1-yl)amino]pyridine-3-carboxamide
2-(ethylamino)-N-[(1R,3S)-3-(4-methylpiperazine-1-carbonyl)cyclopentyl]pyrimidine-5-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(pyrimidin-2-yl)pyrrolidin-3-yl]-3-methanesulfonamidopropanamide
3-(2-chlorophenyl)-1-cyclopentyl-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]pyrrolidine-2,5-dione
2-(1H-pyrazol-1-yl)-1-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)butan-1-one
2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carboxamide
(3aR,7aS)-2-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-(6-aminopyrimidin-4-yl)-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
2-(2,3-dihydro-1H-inden-1-yl)-N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}acetamide
3-methyl-N-(1-{1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
N-[(4-ethylphenyl)methyl]-5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
6-({[4-(dimethylamino)oxan-4-yl]methyl}amino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
4-ethyl-3-(1-{2-[(2-methoxyethyl)(methyl)amino]acetyl}piperidin-3-yl)-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine