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3-[1-(3-oxo-3,4-dihydroquinoxaline-2-carbonyl)piperidin-3-yl]benzoic acid
4-ethyl-3-{1-[(5-ethylpyridin-2-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
{1-[(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methanol
4-{3-oxa-9-azaspiro[5.5]undecan-9-ylmethyl}-1H-pyrazole-3-carboxylic acid
1-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}but-3-en-1-one
N,N-dimethyl-4-[3-(1H-pyrazol-5-yl)phenyl]benzamide
3-[(4-fluorophenyl)methyl]-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine
N-({1-[(2-cyanophenyl)methyl]pyrrolidin-3-yl}methyl)-2-methoxyacetamide
1-[2-(furan-2-yl)azepan-1-yl]-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
(1R,5S,8S)-3-[(5-ethylpyridin-2-yl)methyl]-8-methoxy-3-azabicyclo[3.2.1]octane
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-[1-(oxan-4-yl)piperidine-4-carbonyl]piperidin-4-ol
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-(dimethyl-1,3-thiazol-5-yl)ethan-1-one
3-[2-(dimethylamino)ethyl]-1-ethyl-8-[4-(4-methoxyphenyl)butan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{3-[5-(thiophen-2-yl)furan-2-yl]propanoyl}morpholine-2-carboxylic acid
1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}-3-(2-methoxyphenyl)propan-1-one
4-{2-[1-(4-chlorophenyl)-5-oxo-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetyl}piperazin-2-one
methyl 4-{4-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperazin-1-yl}benzoate
2-phenoxy-N-(1-{7-[(4-phenylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
3-benzyl-N-[1-(2-chlorophenyl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-methyl-2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)-N-{[2-(methylamino)pyrimidin-5-yl]methyl}acetamide
N-({1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}methyl)-5-methylpyrazine-2-carboxamide
(1r,4r)-4-{[2-(3-fluoro-4-hydroxyphenyl)acetamido]methyl}-N-methylcyclohexane-1-carboxamide
4-[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]-N-(3-methoxyphenyl)piperidine-1-carboxamide
3-amino-1-[(5-chloro-2,3-dimethoxyphenyl)methyl]pyrrolidine-3-carboxylic acid
1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(1-methyl-1H-imidazol-2-yl)piperidine
2-({[3-(dimethylamino)thiolan-3-yl]methyl}amino)-N-[(2-methoxyphenyl)methyl]acetamide
1-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-3-methyl-1,2-dihydroquinoxalin-2-one
N-(2-hydroxyethyl)-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
6-{[2-(trifluoromethyl)morpholin-4-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-methoxy-3-methyl-2-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}-1H-indole
4-[4-(1-acetylpiperidine-4-carbonyl)piperazin-1-yl]-2-[(3-fluorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
1-methanesulfonyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]piperidin-4-amine
1-[cyclohexyl(methyl)amino]-3-[3-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenoxy]propan-2-ol
2-ethyl-1-(2-methyl-1-benzofuran-5-carbonyl)-2,5-dihydro-1H-pyrrole
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(phenylsulfanyl)ethan-1-one
2-(2H-1,3-benzodioxol-5-yloxy)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
2-(pyridin-2-yl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-[(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carboxamide
1-ethyl-4-{1-ethyl-5-phenyl-1H-pyrazolo[3,4-b]pyridin-6-yl}-1H-pyrazole
N-benzyl-6-(piperidin-3-yl)-N-(1,3-thiazol-2-ylmethyl)pyrimidin-4-amine
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(morpholin-4-yl)propyl]acetamide
8-[(2S)-2-aminohexanoyl]-2-[(4-chlorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-(1-benzyl-1H-pyrazol-5-yl)-2-{1H-pyrazolo[3,4-b]pyridin-1-yl}acetamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}({[3-(methylsulfanyl)phenyl]methyl})(oxolan-2-ylmethyl)amine
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-2-(propan-2-yl)-1,3-thiazole-4-carboxamide
(butan-2-yl)({[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl})(pyridin-4-ylmethyl)amine
(3aR,6aR)-N-{[2-(benzyloxy)phenyl]methyl}-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-4-carboxamide