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N-(1-{7-[(2-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
(1R,2R,4R)-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-[(2-fluorophenyl)methyl]-N-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
5,7-dimethyl-3-[3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]-[1,2,4]triazolo[4,3-a]pyrimidine
ethyl({[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})(pyridin-4-ylmethyl)amine
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-4-{[5-(hydroxymethyl)furan-2-yl]methyl}-1-(2-methylpropyl)-1,4-diazepan-2-one
2-(4-{[5-(methoxymethyl)furan-2-yl]methyl}-1-(2-methylpropyl)piperazin-2-yl)ethan-1-ol
(furan-2-ylmethyl)({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})amine
5-(3-acetylphenoxymethyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1H-pyrazole-3-carboxamide
N-cycloheptyl-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
1-[1-(propan-2-yl)piperidine-4-carbonyl]-4-(pyridin-3-yl)piperidin-4-ol
2-(4-fluorophenyl)-1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)azetidine
(2S,3R)-2-amino-3-hydroxy-1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]butan-1-one
2-tert-butyl-4-hydroxy-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}pyrimidine-5-carboxamide
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl](1H-imidazol-4-ylmethyl)methylamine
1-(5-ethyl-1,3-oxazole-4-carbonyl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
2-(2-methoxyethyl)-9-[4-(methylsulfanyl)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
(3S,4R)-1-{[3-(difluoromethoxy)phenyl]methyl}-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
(1R,7S)-3-cycloheptyl-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-oxo-2-(pyridin-3-yl)acetamide
methyl[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
(4aR,7aS)-1-(3-methylbutanoyl)-4-(1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(1H-pyrrol-1-yl)ethyl]benzamide
N-{1-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
(3R,4S)-4-cyclopropyl-1-[6-(piperidine-1-carbonyl)pyrazin-2-yl]pyrrolidin-3-amine
1-(4-{[2-(2-hydroxyethoxy)ethyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-[(3S,4R)-1-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
4-[1-({2-[(dimethylamino)methyl]phenyl}methyl)-4-phenyl-1H-imidazol-5-yl]-2-methoxyphenol
9-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-oxa-9-azaspiro[5.5]undecane
N-(2-{7-[(4-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methylbenzamide
N-[2-(azepan-1-yl)ethyl]-N-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
N-[3-(5-chloro-1H-1,3-benzodiazol-2-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
4-cyclohexyl-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
8-(1-methoxypropan-2-yl)-1-methyl-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(1,3,4-thiadiazol-2-yl)pyrrolidin-3-yl]methanol
1-methyl-3-(2-methylpropyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-6-(2-methylphenyl)-N-[1-(pyridin-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-benzyl-N,N-dimethyl-4-(2-methylphenyl)-5-oxopiperazine-1-sulfonamide
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(furan-2-ylmethyl)piperidine
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
5-(cyclohexylmethyl)-7-{[(oxolan-2-ylmethyl)amino]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
1-[1-(3-ethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-3-phenylpropan-1-ol
1-(5-methyl-1,3,4-thiadiazol-2-yl)-4-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperazine
8-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-1-oxa-8-azaspiro[4.6]undecane
4-(2-methylpropanoyl)-1-(2-phenylphenyl)piperazin-2-one
4-[5-(4-chloro-1-methyl-1H-pyrazol-3-yl)-1-cyclohexyl-1H-1,2,4-triazol-3-yl]pyridine