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2-cyclopropyl-N-(3,4-difluorophenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
8-(1,3-benzothiazol-2-ylmethyl)-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[1-(6-cyanopyridin-2-yl)piperidin-3-yl]methyl}-2-(2-methoxyphenoxy)acetamide
N-[2-(6-methylpyridin-2-yl)ethyl]-5-(naphthalen-2-yl)-1,2,4-triazin-3-amine
({4-cyclopropyl-5-[1-(pyrazin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-8-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(3,4-dimethylpiperazin-1-yl)-5-(3-fluoro-4-methoxyphenyl)-1,2,4-triazine
4-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2,6-dimethylpyrimidine
5-(2-methoxyacetamido)-N-methyl-1-(2-phenylethyl)-N-[2-(1H-pyrazol-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
4-methoxy-1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-4-phenylpiperidine
1-(2,3-dimethylphenyl)-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}piperidine
5-methoxy-1-methyl-2-[(2S)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl]-1H-indole
N-methyl-2-[methyl(phenyl)amino]-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
3-(oxolan-2-yl)-7-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-[2-({[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}methyl)phenoxy]acetic acid
N-(2-methoxyethyl)-3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)propanamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1-ethylpiperidin-4-yl)pyrrolidin-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
(4S,6R)-N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-6-methyl-2-sulfanylidene-1,3-diazinane-4-carboxamide
8-[(8-chloroquinolin-2-yl)methyl]-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1s,4s)-4-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclohexan-1-ol
2-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidine-1-carbonyl]thiophen-3-amine
3-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]pyridin-2-amine
2-chloro-N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}pyridine-4-carboxamide
1-(cyclohexylmethyl)-N5-[(1R)-1-(3-methoxyphenyl)ethyl]-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-methyl-6-oxo-N-(pentan-3-yl)-N-(2-phenylethyl)-1,6-dihydropyrimidine-5-carboxamide
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
2-[2-(1H-imidazol-4-yl)ethyl]-9-(2-methyloxolane-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazole-3-carboxamide
4-[(2-chloro-4,5-diethoxyphenyl)methyl]-2-(trifluoromethyl)morpholine
(1S,2S,9S)-6-oxo-N-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-7,11-diazatricyclo[7.3.1.02,7]tridecane-11-carboxamide
4-(5-chloropyrimidin-2-yl)phenol
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-methyl-1,3-thiazole-5-carbonyl)piperidine
methyl (2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-{[2-(3-methylpyridin-2-yl)ethyl]carbamoyl}pyrrolidine-2-carboxylate
1-(1-benzofuran-5-ylmethyl)-4-(3,4-difluorophenoxy)piperidine-4-carboxylic acid
3-[2-(3-chloro-5-fluoro-4-methoxyphenyl)-1H-imidazol-1-yl]pyrrolidin-2-one
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamide
N-tert-butyl-2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}acetamide
[3-(2-methoxyethyl)-1-(pyrimidin-2-yl)piperidin-3-yl]methanol
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-ethylphenyl)methyl]-N-methylacetamide
2-(2-hydroxyethyl)-8-[(2-methoxy-3,5-dimethylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-hydroxy-3-[(4-hydroxypiperidin-1-yl)methyl]-1-(3-phenylpropyl)piperidin-2-one
{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(ethyl)(pyridin-4-ylmethyl)amine
2-butyl-4-({4-cyclopropyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1H-imidazole
5-methyl-4-({2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}amino)thieno[2,3-d]pyrimidine-6-carboxylic acid
3,6,7-trimethyl-N-[2-(6-methylpyridin-2-yl)ethyl]-1-benzofuran-2-carboxamide
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]ethan-1-one
3-[ethyl(pyridin-4-ylmethyl)amino]-N-(2-phenylphenyl)piperidine-1-carboxamide
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-2-(methylsulfanyl)acetamide
N3-cyclohexyl-1-(2-methylpropyl)-4-oxo-N5-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide