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3-methyl-1-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pentane-1,2-dione
1-benzyl-8-(2,2-dimethylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2,4-dimethoxyphenyl)-3-[1-(oxolan-3-ylmethyl)piperidin-4-yl]propanamide
methyl 1-[(3R,5S)-1-cyclohexyl-5-{[2-(1H-indol-3-yl)ethyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(1S,5R)-3-(3-phenylpropyl)-6-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-3-phenylprop-2-ynamide
1-cyclohexyl-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-1H-1,2,3-triazole-4-carboxamide
N-{[7-(1,3-benzothiazol-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,2-dimethyloxane-4-carboxamide
4-(1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-imidazol-2-yl)pyridine
(2S)-N,N-dimethyl-1-{[4-(6-oxo-4-propyl-1,6-dihydropyrimidin-2-yl)phenyl]methyl}pyrrolidine-2-carboxamide
4-ethyl-N-(2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-oxoethyl)cyclohexane-1-carboxamide
1-(1H-imidazol-4-ylmethyl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
(3R,4R)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-3-cyclopropyl-4-methylpyrrolidin-3-ol
1-(2-methoxyethyl)-8-[4-(4-methoxyphenyl)butan-2-yl]-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[2-(2,4-dimethylphenoxy)ethyl](methyl)(pyridin-4-ylmethyl)amine
8-methoxy-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(morpholin-4-yl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-2-(pyridin-3-yl)acetamide
methyl 2-[4-(8-fluoroquinoline-2-carbonyl)-3-methyl-2-oxopiperazin-1-yl]acetate
N-cyclopropyl-3-methoxy-N-[(7-methoxy-2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}quinolin-3-yl)methyl]benzamide
methyl({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)(pyridin-2-ylmethyl)amine
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[(1-phenylcyclopentyl)methyl]benzamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
methyl 3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl]propanoate
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-ol
4-(1-methyl-1H-imidazol-2-yl)-1-[2-(phenylsulfanyl)ethyl]piperidine
3-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperidine-3-carbonyl]pyridine
ethyl 2-{[3-({[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}carbamoyl)phenyl]amino}acetate
2-(2-{[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
3-methyl-1-[4-(2-methylpropyl)-1,4-diazepan-1-yl]but-2-en-1-one
5-methyl-3-({3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidin-1-yl}methyl)-1H-indole
2-[4-(cyclohexylmethyl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
1-[4-(3,6-dimethylpyrazin-2-yl)-6-hydroxy-1,4-diazepan-1-yl]ethan-1-one
3-(1-methyl-1H-imidazol-2-yl)-6-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}pyridazine
N-[(4-hydroxyphenyl)methyl]-2-(propan-2-yloxy)-N-(pyridin-4-ylmethyl)propanamide
methyl 2-(cyclopentylsulfamoyl)-6-(4-phenylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-amino-4-(4-cyanophenyl)-6-(4-hydroxyphenyl)-5-methylpyridine-3-carbonitrile
methyl 3-(cyclobutylmethoxy)-5-{methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]carbamoyl}benzoate
8-(1H-indol-2-ylmethyl)-1-(2-methoxyethyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 1-(3-phenylpropyl)-5-(1H-pyrazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[(3-cyanophenyl)methyl]-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}[2-(1H-imidazol-1-yl)ethyl]methylamine
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]acetamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-3-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
N-{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}cyclopentanamine
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]benzamide
6-[2-({1,9-dioxaspiro[5.5]undecan-4-yl}amino)ethyl]-2-methylpyrimidin-4-ol
4-hydroxy-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinolin-2-yl}piperidine-4-carboxylic acid
3-(4-ethylphenyl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1H-pyrazole-5-carboxamide
5-(4-benzoylpiperidine-1-carbonyl)-4,6-dimethyl-1,2,3,4-tetrahydropyrimidin-2-one