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N-[2-(dimethylamino)ethyl]-3-[1-(thiolan-3-yl)piperidin-4-yl]propanamide
methyl 2-{[3-(2-phenylacetyl)piperidine-1-carbonyl]amino}acetate
1-(3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-oxopropyl)azepan-2-one
2,3-dimethyl-6-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}quinoxaline
N-({3-methyl-7-[3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-2-yl)acetamide
1-[(2-chloro-6-fluorophenyl)methyl]-3-cyclopentyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-1H-1,2,4-triazole
2-[4-(hydroxymethyl)phenyl]-1-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}ethan-1-one
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
(2S,4R)-N,N-diethyl-4-{4-[(2-hydroxyethyl)(methyl)amino]benzamido}-1-methylpyrrolidine-2-carboxamide
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N,2-dimethyl-2,8-diazaspiro[4.5]decane-3-carboxamide
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
4-hydroxy-2-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)quinoline-6-carboxamide
1-(4-fluorophenyl)-4-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)piperazine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
2-cyclopentyl-8-(2,6-dimethylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-(pyridin-2-ylmethyl)-1-[1-(1,3-thiazol-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(2R,6R)-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-hydroxy-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)benzamide
3-{2-[1-methyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-indole
2-(4-chlorophenyl)-4-[2-(1H-1,2,4-triazol-3-yl)benzoyl]morpholine
N-{2-[4-(furan-2-ylmethyl)morpholin-2-yl]ethyl}cyclopropanesulfonamide
6-methoxy-3-{[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
2-(morpholin-4-yl)-8-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methoxy}quinoline
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[(3R)-3-fluoropyrrolidin-1-yl]acetamide
3-(1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)-1-(morpholin-4-yl)propan-1-one
1-(1-cyclobutylpiperidin-3-yl)-4-(4-fluorophenyl)piperazine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[2-(4-fluorophenyl)pyrrolidin-1-yl]butan-1-one
ethyl 4-[1-(1,3-dioxo-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindol-4-yl)piperidine-4-carbonyl]piperazine-1-carboxylate
N-{2-[benzyl(methyl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl}-1-hydroxycyclopentane-1-carboxamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-N-(2-methoxyethyl)-5-methyl-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl})methylamine
4-methyl-2-(1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-1H-1,3-benzodiazole
5-chloro-6-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]pyridine-3-carboxylic acid
4-[2-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-oxoethyl]-5-methyl-2,3-dihydro-1H-pyrazol-3-one
3-(2-{[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]amino}ethyl)-1,3-oxazinan-2-one
1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(1-methyl-1H-imidazol-2-yl)piperidine
(2S)-2-amino-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-4-(methylsulfanyl)butan-1-one
2-{8-[(4-methoxyphenyl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
5-({[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}sulfanyl)-1H-1,2,4-triazol-3-amine
ethyl 1-({5-[(adamantan-2-ylmethyl)carbamoyl]-6-oxo-1,6-dihydropyridin-2-yl}methyl)piperidine-4-carboxylate
{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}(methyl)(1H-pyrazol-3-ylmethyl)amine
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 2-[1-(2-methoxyethyl)-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
propan-2-yl 4-chloro-3-({[(3-methyloxetan-3-yl)methyl]carbamoyl}amino)benzoate
3-(1H-imidazol-1-yl)-1-[4-(4-methoxybenzoyl)piperazin-1-yl]butan-1-one
N6-(2-methoxyethyl)-N5-methyl-N5-[2-(pyrrolidin-1-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
5-(quinolin-8-yl)-2,3-dihydro-1H-inden-1-one
2-methoxy-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)benzamide
N-[1-(1-cyclobutanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-4-phenylbutanamide