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N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)cyclopropanamine
1-(carbamoylmethyl)-N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]piperidine-4-carboxamide
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
N-[(2-ethoxypyridin-3-yl)methyl]-2-methyl-3-[(pyridin-2-ylmethyl)amino]benzamide
N-[2-(adamantan-1-yl)propan-2-yl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
5,7-dimethyl-N-[(2-phenoxypyridin-3-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
4-{3-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
{4-[(3-fluorophenyl)methyl]-1-[(E)-2-phenylethenesulfonyl]piperidin-4-yl}methanol
4-{[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
6-ethyl-2-oxo-N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1,2-dihydropyridine-4-carboxamide
1-[(1-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(4,6-dimethyl-1-benzofuran-3-yl)ethan-1-one
5-(3-fluoro-4-methoxyphenyl)-N-(oxan-4-ylmethyl)-1,2,4-triazin-3-amine
1-(2-{[3-(3-methoxyphenyl)-1H-pyrazol-4-yl]formamido}ethyl)piperidine-3-carboxamide
[(3S,5R)-1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
2-[2-(dimethylamino)acetyl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-amino-N-{[2-(dimethylamino)pyridin-3-yl]methyl}-6-(2-methylpropyl)pyrimidine-4-carboxamide
3-[1-(4-chloro-3-fluorobenzoyl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(4-ethoxyphenyl)-5-(methoxymethyl)-3-methyl-1H-pyrazole
2-[1-butyl-3-(2-methylbutyl)-1H-1,2,4-triazol-5-yl]ethan-1-ol
5-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-5-(2-methylpropyl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
2-[5-(1-benzyl-1H-pyrazol-4-yl)-1-cyclohexyl-1H-1,2,4-triazol-3-yl]acetamide
3-chloro-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)benzamide
({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)(methyl)(pyridin-3-ylmethyl)amine
3-{5-[(phenylsulfanyl)methyl]-1H-1,2,4-triazol-3-yl}pyridine
methyl 5-[(butan-2-yl)amino]-3-(2-methylbutanamido)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
methyl 4-({4-[(2-fluorophenyl)methyl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylate
({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-(cyclohexylmethyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
(2R,3S,6R)-5-(4-fluorobenzoyl)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(3-methylbutyl)-5-{1-[5-(propan-2-yl)pyrimidin-4-yl]piperidin-4-yl}imidazolidine-2,4-dione
2-[1-(7-fluoro-3-methyl-1H-indole-2-carbonyl)pyrrolidin-2-yl]-6-methyl-1H-1,3-benzodiazole
N-cyclopropyl-2-ethyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)butanamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
(4S,4aS,8aS)-1-(dimethyl-1,2-oxazole-4-carbonyl)-4-phenyl-decahydroquinolin-4-ol
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N,2-diethylpyrimidine-5-carboxamide
(3R)-1-({2-[4-(morpholin-4-yl)butoxy]phenyl}methyl)pyrrolidin-3-ol
5-[1-(2,3-dihydro-1H-inden-2-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]pyrazin-2-ol
N-butyl-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-(2-phenoxyethyl)piperidin-4-yl}methanol
1-[(4-chlorophenyl)methyl]-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(2-methoxyphenoxy)ethan-1-one
5-(3-methoxyphenyl)-3-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}-1,2,4-triazine
3-{5-[(4-fluoro-3-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
[1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-2-yl]methanol
(1S,5R)-6-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-phenyl-5-[2-(propan-2-ylsulfanyl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide