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methyl 3-(4-tert-butylbenzoyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-4-methylbenzamide
N-(1-methylpiperidin-4-yl)-2-(morpholin-3-yl)-N-(2-phenylethyl)acetamide
1,5,6-trimethyl-2-oxo-N-{2-[2-(trifluoromethyl)phenyl]ethyl}-1,2-dihydropyridine-3-carboxamide
1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
3-(3-hydroxyphenyl)-3-(4-hydroxyphenyl)-1-(piperidin-1-yl)propan-1-one
ethyl 4-[(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)methyl]-1H-pyrazole-3-carboxylate
3-{2-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]phenyl}-1H-1,2,4-triazole
1-{5-[(2S)-2-(3-ethyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-2-methylphenyl}imidazolidin-2-one
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-3-fluorobenzamide
N-butyl-N-methyl-3-{[({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)amino]methyl}imidazo[1,2-a]pyridine-2-carboxamide
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
1-{1'-[(4-ethoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
1-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}azetidin-3-ol
3-{1-[1-(2-aminoacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea
5,8-dimethyl-2-({[1-(pyrazin-2-yl)propan-2-yl]amino}methyl)quinolin-4-ol
{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
3-{[4-(1-benzofuran-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
ethyl 4-[(4-chlorophenyl)methyl]-1-(1-methylazepane-2-carbonyl)piperidine-4-carboxylate
2-(2-chloro-4-fluorophenoxymethyl)-N-[2-(pyridin-3-yl)ethyl]-1,3-oxazole-4-carboxamide
3,5-dimethoxy-N-{[1-(1,2-oxazol-3-ylmethyl)piperidin-3-yl]methyl}benzamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-({[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
1-(6-methyl-2-propylpyrimidin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-methyl-4-{[1-(2-phenylethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,4-diazepane
2-(1H-indazol-1-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
3-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(2,5-dimethoxyphenyl)-3-propyl-4H-1,2,4-triazole
N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]quinoxaline-5-carboxamide
1-(2-fluoro-4-methanesulfonylphenyl)-4-(1H-1,2,3-triazole-5-carbonyl)piperazine
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[2-(pyridin-3-yloxy)propyl]propanamide
4-[2-(aminomethyl)phenyl]-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
2-methyl-3-[2-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]phenol
7-(cyclobutylmethyl)-2-(4-methylpiperazine-1-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-[(isoquinolin-5-yloxy)methyl]-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1,2-oxazole-3-carboxamide
N-(3,4-dimethylphenyl)-1-(isoquinoline-3-carbonyl)piperidin-3-amine
(propan-2-yl)({[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl})[(trimethyl-1H-pyrazol-4-yl)methyl]amine
5-methyl-1-propyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1H-pyrazole-4-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)piperidin-2-one
6-(2,5-dimethoxyphenyl)-2-(4-methylpiperazin-1-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}pyridine-3-carboxamide
[(3R,4R)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
2-[(2-hydroxyethyl)({[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
2-(cyclohexylmethyl)-4-(5-methyl-1H-pyrazole-3-carbonyl)morpholine
2-(2-acetylbenzoyl)-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one
1-cyclopentyl-N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
(3aR,6aS)-5-[(2,3-difluoro-6-methoxyphenyl)methyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
[2-ethoxy-5-({[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})amino}methyl)phenyl]methanol
4-{4-[1-(isoquinolin-1-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}butanamide
N-(2-{7-[(2,6-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
2-butyl-8-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one