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2-(2H-1,3-benzodioxol-5-yl)-8-methoxy-5-(pyridin-4-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
(2S)-2-({2-[(2,6-dichlorophenyl)methyl]-4-hydroxypyrimidin-5-yl}formamido)propanamide
methyl (2S,4S,5R)-5-(2,3-difluorophenyl)-1-methyl-4-{[2-(pyridin-4-yl)ethyl]carbamoyl}pyrrolidine-2-carboxylate
1-(2-cyclohexylethyl)-3-{[(furan-3-ylmethyl)amino]methyl}-3-hydroxypiperidin-2-one
4-{4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperazin-1-yl}-2,5-dimethylpyrimidine
ethyl 3-benzyl-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxylate
5-(1,2,3,4-tetrahydroisoquinolin-5-yl)-1,2-dihydropyridin-2-one
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-methoxyethan-1-one
(2-{2-[1-(2-methoxypyridine-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
6-ethyl-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-methylquinoline-4-carboxamide
2-{[5-(2-chlorophenyl)furan-2-yl]formamido}-4-(methylsulfanyl)butanoic acid
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2,6-dimethoxypyridine-3-carboxamide
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-(4-propanoylphenoxy)acetamide
2-(1-{imidazo[1,2-b]pyridazine-3-carbonyl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
(2S)-2-amino-N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-(methylsulfanyl)butanamide
(2R)-2-amino-1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
1-methyl-6-(pyridin-3-yl)-N-[1-(thiophen-3-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
3-(1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carbonyl)pyridine
N-methyl-N-[(5-methylfuran-2-yl)methyl]-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
2-{4-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]piperidin-1-yl}acetamide
6-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]amino}-N,N-dimethylpyrazine-2-carboxamide
3-methyl-7-(quinoxaline-5-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-(azepan-1-yl)-3-[(pyrimidin-2-yl)amino]propan-2-ol
2-{4-[(2,4-dimethyl-3-oxopiperazin-1-yl)methyl]phenyl}-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
N-{1-[1-(cyclobutylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
N-{[5-chloro-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,6-difluorobenzamide
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
methyl[(1-methyl-1H-pyrazol-4-yl)methyl]{[4-({1-[4-(trifluoromethyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}amine
5-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-methyl-N-(3-phenylprop-2-yn-1-yl)-N-propyl-1H-1,2,3-benzotriazole-5-carboxamide
6-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-(2-methoxyphenyl)-5-(quinolin-5-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
(1S,5R)-3-methyl-6-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-3,6-diazabicyclo[3.2.2]nonane
{1-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-3-(cyclopropylmethyl)piperidin-3-yl}methanol
2-amino-N-[3-(1H-imidazol-1-yl)propyl]-4-phenylpyrimidine-5-carboxamide
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-(3-hydroxypiperidin-1-yl)ethan-1-one
4-(3-acetylbenzoyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
{2-[2-benzyl-4-(3-methoxyphenyl)-5-oxopiperazin-1-yl]-2-oxoethyl}urea
[(3R,5R)-1-(4-phenylbenzoyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
5-{6-chloro-2-methylimidazo[1,2-a]pyridine-3-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-[3-({[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amino}methyl)-1H-indol-1-yl]acetamide
(3R,4R)-1-[(dimethyl-4H-1,2,4-triazol-3-yl)methyl]-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
2-(4-ethyl-3,3-dimethylpiperazin-1-yl)-2-(5-fluoro-2-methoxyphenyl)acetic acid
1-(cyclopropylmethyl)-4-[(4-methanesulfonylphenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
N-[(3R,4R)-1-(6-cyanopyridin-2-yl)-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](methyl){[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
1-[2-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-(1-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide