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3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-(1,3-dihydroxy-2-methylpropan-2-yl)propanamide
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}piperidin-4-ol
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-2-(1H-indol-3-yl)-N-(2-methoxyethyl)acetamide
1-(4,7-dimethylquinazolin-2-yl)-N-(2-phenylpropyl)piperidine-4-carboxamide
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
N,1,3-trimethyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-(propan-2-yl)-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}piperidine-3-carboxamide
4-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1-(prop-2-en-1-yl)pyrrolidin-2-one
2-[1-(5-chloro-2-methoxyphenyl)-5-[1-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
4-chloro-5-{[({3-[(dimethylamino)methyl]phenyl}methyl)(methyl)amino]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-1-ethyl-1H-pyrazole-4-carboxamide
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(thiophen-2-yl)ethyl]acetamide
2-(2,3-dihydro-1H-isoindol-2-yl)-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
(3R,4R)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-(pyridin-4-ylmethyl)piperidin-3-ol
2-(2-methoxyethyl)-N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-1,3-benzoxazole-6-carboxamide
methyl 4-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}benzoate
4-(3-phenylpropyl)-7-{[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-methyl-3-[2-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
(3aS,6aS)-2-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[2-(trifluoromethyl)phenyl]urea
1-methyl-N-(1-phenylbutyl)-1H-pyrrole-2-carboxamide
4-{3-cyclopropyl-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-5-methyl-1-propyl-1H-pyrazole
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}acetamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-4-yl]propanamide
2-methoxy-4-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]pyridine-3-carbonitrile
4-{1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-1H-pyrazole-4-carbonyl}piperazine-1-carbaldehyde
2-(3-{[3-(aminomethyl)piperidin-1-yl]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
4-{1-[4-(difluoromethoxy)phenyl]-1H-imidazol-2-yl}-3-methoxyphenol
2-[(furan-3-ylmethyl)amino]-N-[2-(2-methoxyphenyl)ethyl]acetamide
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
5-fluoro-3-methyl-2-{[3-(pyridin-2-yl)azetidin-1-yl]methyl}-1H-indole
1-(4-methoxybenzoyl)-4-(2-methyl-1,3-thiazole-5-carbonyl)piperazine
2-[3-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)-1H-indol-1-yl]acetamide
4-{4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-[(1S,5R)-6-(3,5-dimethoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(1S,5R)-3-(pyridin-3-ylmethyl)-6-[3-(trifluoromethyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
2-{4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]morpholin-3-yl}-N-(pyridin-3-yl)acetamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-(propan-2-yl)propanamide
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-[(1-benzylpiperidin-4-yl)methyl]-1-(methoxymethyl)-N-methylcyclobutane-1-carboxamide
4-[(5-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
methyl 5-[(1-acetylpiperidin-4-yl)amino]-3-(2-methoxyacetamido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-benzyl-8-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-2,8-diazaspiro[4.5]decan-3-one
1-{3-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-3-oxopropyl}azepan-2-one
6-(4-ethylphenyl)-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3,6-dimethyl-N-[2-(1,3-thiazol-4-yl)ethyl]-1-benzofuran-2-carboxamide
1-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]-4-(4-methoxyphenyl)butan-1-one
ethyl 1-{[3-(2-hydroxyethoxy)phenyl]methyl}-4-(2-phenoxyethyl)piperidine-4-carboxylate
4-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-4-oxobutane-1-sulfonamide