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N-[3-(1,3-thiazol-4-yl)phenyl]-1H-indazole-3-carboxamide
N-(3-chloro-4-fluorophenyl)-N'-methyl-N'-[1-(pyridin-3-yl)ethyl]butanediamide
1-[(3,4-difluorophenyl)methyl]-3-({[(4-fluorophenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
N-[(2-chloro-6-fluorophenyl)methyl]-N-ethyl-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-(prop-2-en-1-yl)-5-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
1-benzyl-5-(pyridine-3-carbonyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[benzyl(methyl)amino]-3-[4-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]-4-(thiophen-2-yl)butan-1-one
6-(2-butoxy-4-fluorophenyl)-N,N-dimethylpyridazin-3-amine
1-{3-[1-cyclohexyl-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]phenyl}imidazolidin-2-one
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N,6-dimethyl-2-(pyridin-3-yl)pyrimidin-4-amine
5-(2,4-difluorophenoxymethyl)-N-(thiophen-3-ylmethyl)-1H-pyrazole-3-carboxamide
N-{1-[4-(3-chlorophenyl)-5-({[3-(trifluoromethyl)phenyl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}pyridine-2-carboxamide
6-(2-chlorophenyl)-N-(1-hydroxy-3-methylbutan-2-yl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
methyl[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[(4-methoxyphenyl)methyl]propanamide
3-{2-[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-oxoethyl}-4-(propan-2-yl)piperazin-2-one
3-(1-methyl-1H-pyrazol-4-yl)-N-[(5-methylpyrazin-2-yl)methyl]propanamide
N-(1-cycloheptylpiperidin-3-yl)-4-(methylsulfanyl)benzamide
methyl({[3-(methylsulfanyl)phenyl]methyl}){[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}amine
2-{[4-(2,3-difluoro-4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
(3R,4R)-1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-benzyl-3-(4-methyl-1,3-thiazol-5-yl)-N-[(6-methylpyridin-2-yl)methyl]propanamide
2-(pyridin-3-yl)-1-{4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}ethan-1-one
5-[3,6-dimethyl-4-(pyrrolidine-1-carbonyl)quinolin-2-yl]-N-ethylpyrimidin-2-amine
N-[1-(quinolin-5-ylmethyl)piperidin-3-yl]acetamide
(1S,5R)-6-(cyclopropylmethyl)-3-[3-oxo-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopentyl-5-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(dimethylamino)-2-[3-(4-fluorophenoxy)propyl]-2,3-dihydropyridazin-3-one
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-(quinolin-8-ylmethyl)piperidin-3-ol
3-{imidazo[1,2-a]pyridin-2-yl}-N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
2-(4-cyclohexylpiperazin-1-yl)-2-[4-(dimethylcarbamoyl)phenyl]acetic acid
5-{3-oxo-3-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propyl}imidazolidine-2,4-dione
N-[(5-{[(1s,4s)-4-aminocyclohexyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]cyclobutanecarboxamide
1-(cyclopropylmethyl)-5-(quinoline-8-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
7-methoxy-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{1-cyclopentyl-4-[(2-methyl-1H-imidazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
4-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-1-(pyrrolidine-1-carbonyl)piperidine
4-chloro-N-[(4-hydroxyazepan-4-yl)methyl]-2,5-dimethylbenzene-1-sulfonamide
N-[(2,3-dimethoxyphenyl)methyl]-4-methyl-5-{1-[3-(6-methylpyridin-2-yl)propyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
4-methoxy-3-{[2-(trifluoromethyl)morpholin-4-yl]methyl}phenol
1-[(3-{[1-(furan-3-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-methyl-1,4-diazepane
N,N-dimethyl-4-(1-{[(2-methyl-2H-1,2,3-triazol-4-yl)carbamoyl]methyl}-1H-indol-5-yl)benzamide
4-(4-benzylpiperazin-1-yl)-2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}propanamide
N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]thiolan-3-amine
2-{[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]amino}-N-(4-methylphenyl)propanamide