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(3S,4R)-3-ethyl-1-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-4-methylpiperidin-4-ol
1-[4-(2-{1-oxa-8-azaspiro[4.5]decan-8-yl}-2-oxoethyl)phenyl]imidazolidin-2-one
N-(2-methoxyethyl)-N-methyl-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(5-ethyl-1,3-oxazole-4-carbonyl)spiro[azepane-4,2'-chromene]
4-(pyridin-4-ylmethyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclobutanecarboxamide
methyl 6-(cyclohex-3-ene-1-carbonyl)-2-{[(2-fluorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-4,6-dimethylpyridine-3-carboxamide
N-[(5-chloro-2-methoxyphenyl)methyl]-N-methyloxolane-3-carboxamide
2-amino-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
1-(4-methylpiperidin-1-yl)-3-[(3S,4R)-1-(propan-2-yl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propan-1-one
9-ethyl-1-methyl-4-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(pent-2-yn-1-yl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
1-{2-[2-(4-fluorophenyl)-1H-imidazol-1-yl]ethyl}azepane
1-[2-(dimethylamino)ethyl]-N-[2-(2-methoxynaphthalen-1-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
5-[1-(4-methylquinolin-2-yl)piperidin-4-yl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
N-[1-(2,4-dimethylphenyl)propyl]-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(3-methoxypropyl)-1-[(4-methylthiophen-2-yl)sulfonyl]piperidine
4-[(2-methylpyridin-3-yl)oxy]-1-(1,3-thiazol-2-yl)piperidine-4-carboxylic acid
3-{1-[(3-methyl-1-benzofuran-2-yl)methyl]-1H-imidazol-2-yl}pyridine
N-{1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1-oxopentan-2-yl}acetamide
5-(2H-1,3-benzodioxol-5-yl)-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1,2,4-triazin-3-amine
2-(adamantan-1-yl)-5-[4-(methylamino)piperidine-1-carbonyl]pyrimidin-4-ol
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(methylamino)-1,3-thiazole-4-carboxamide
3-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-[4-(oxan-2-ylmethoxy)phenyl]urea
2-methyl-2-{[5-(4-phenylazepane-1-carbonyl)pyridin-2-yl]amino}propane-1,3-diol
N-[(1-ethylpyrrolidin-2-yl)methyl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
1-(carbamoylmethyl)-N-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-methylpropyl]piperidine-4-carboxamide
2-methoxy-1-[4-(5-propyl-1,2-oxazole-3-carbonyl)-1,4-diazepan-1-yl]ethan-1-one
1-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
(5-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}furan-2-yl)methanol
1-(4-methoxyphenyl)-3-methyl-4-(quinoline-3-carbonyl)piperazin-2-one
2-cyclopropyl-6-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1,3-benzoxazole
N-cyclopentyl-6-(3,4-dimethylpiperazin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-[(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetic acid
(3R,4S)-4-{4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1,4-diazepan-1-yl}oxolan-3-ol
4-[(1-ethyl-1H-pyrazol-3-yl)methyl]-6-fluoro-3,4-dihydro-2H-1,4-benzoxazin-3-one
[(3R,4R)-1-(2,6-dimethoxybenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-[1-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)piperidin-3-yl]benzoic acid
3-benzyl-4-(3,5-difluorobenzoyl)piperazin-2-one
2-(1,3-benzothiazol-2-ylmethyl)-4-[4-(4-phenylpiperazine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
6-ethoxy-2-{[3-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}quinoline
3-({1-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-1,2,3-triazol-4-yl}methyl)-2,3-dihydro-1,3-benzoxazol-2-one
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
4-[3-(cyclopropylmethyl)-5-[4-(1H-imidazol-1-yl)phenyl]-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
N-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-4-(pyridin-4-yl)piperidine-1-carboxamide
4-[4-(cyclohexylmethyl)-1H-1,2,3-triazol-1-yl]-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine
4-[(4-fluorophenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
2-(3,5-dimethylfuran-2-carbonyl)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane