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N-{[1-(quinolin-2-ylmethyl)pyrrolidin-3-yl]methyl}cyclopropanesulfonamide
N-[2-(1-benzylpyrrolidin-3-yl)ethyl]-2-cyclopropylpyrimidine-5-carboxamide
1-{1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
ethyl 2-[(3-{[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)carbamoyl}phenyl)amino]acetate
1-(4-carboxy-1,3-oxazol-2-yl)-3-(2-phenoxyethyl)piperidine-3-carboxylic acid
5-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-N-cyclopentyl-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3S,4S)-1-(benzenesulfonyl)-4-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]pyrrolidin-3-ol
N-[(2,5-difluorophenyl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{1-[(4-phenoxyphenyl)methyl]piperidin-3-yl}propanamide
(2R)-2-amino-N-methyl-2-phenyl-N-(thiophen-3-ylmethyl)acetamide
(3S)-3-ethyl-4-[4-(1H-pyrazol-1-yl)benzenesulfonyl]morpholine
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
4-({4-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]furan-2-yl}methyl)morpholine
1-({1-[2-(azocan-1-yl)acetyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
methyl 6-[2-(2-fluorophenyl)acetyl]-2-[(2-methylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N5-(cyclohexylmethyl)-N3-methyl-4-oxo-N3-(2-phenylethyl)-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(2-hydroxyethyl)-1-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-3-yl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
1-[(4-phenyl-1,3-thiazol-2-yl)methyl]-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
N-[2-(7-methyl-1H-indol-3-yl)ethyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-[(5-ethylpyridin-2-yl)methyl]-4-hydroxy-N-methyl-2-(4-methylphenyl)pyrimidine-5-carboxamide
1-(2-{[benzyl(methyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-methyl-3-phenyl-8-(pyridine-3-carbonyl)-1,8-diazaspiro[4.5]decane
N-(1-ethyl-5-oxopyrrolidin-3-yl)-3-(pyrrolidine-1-sulfonyl)benzamide
N-cyclohexyl-2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
(3S,4S)-4-(morpholin-4-yl)-1-(3-propyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-ol
1-ethyl-N-[2-(1H-imidazol-4-yl)ethyl]piperidine-4-carboxamide
1-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-5-phenylpentan-1-one
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]amine
2-{3-cyclopropyl-5-[3-(morpholin-4-yl)propyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-{4-[4-(piperidin-1-yl)piperidine-1-carbonyl]-5-(propan-2-yl)-1H-pyrazol-1-yl}-4-(thiophen-2-yl)pyrimidine
5-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-phenylfuran-3-carboxamide
2-{[(2,5-difluorophenyl)methyl]amino}-N-[1-(4-methylphenyl)ethyl]acetamide
2-(2-hydroxyethyl)-6-{2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetyl}-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
1-cyclopentyl-4-{[(6,7-dimethoxy-4-methylquinolin-2-yl)amino]methyl}pyrrolidin-2-one
N-[(6-methoxy-2H-chromen-3-yl)methyl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-1,3-benzothiazole-6-carboxamide
5-ethyl-2-{3-[1-(pyridin-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-6-(pyrrolidine-1-carbonyl)pyrazin-2-amine
2-methoxy-4-{[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]amino}pyridine-3-carbonitrile
5-cyclopropyl-4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-3-methyl-1H-pyrazole
6-{2-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-2,3-dihydropyridazin-3-one
N-cyclopropyl-3-[5-(2,6-dimethylpyrimidine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
6-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(4-aminopyridin-2-yl)-N-tert-butylbenzene-1-sulfonamide
(3aS,6aS)-2-(2-methoxyethyl)-5-[(3-methyl-1H-indol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{1,4-dioxa-8-azaspiro[4.5]decan-8-yl}-N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-oxobutanamide
3-[4-methoxy-3-(methoxymethyl)benzoyl]-3,9-diazaspiro[5.6]dodecan-10-one
3-(2-amino-1,3-thiazol-4-yl)-N-[(1S,2R)-2-(cycloheptylamino)cyclobutyl]propanamide
3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-1-(2,3,4-trifluorophenyl)urea
3-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide