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8-(1H-pyrazol-3-yl)quinolin-4-amine
2-(2H-1,3-benzodioxol-5-yl)-1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]ethan-1-one
1-(4-fluorophenyl)-4-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]butane-1,4-dione
3,5-dimethoxy-2-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)benzoic acid
N-{[2-(4-acetylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl}-4-methoxy-N-(2-methoxyethyl)benzamide
{3-[(2-methylphenyl)methyl]-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methanol
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-2-(1H-pyrazol-1-yl)acetamide
N-(1H-imidazol-2-ylmethyl)-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-2-amine
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-3-(1H-imidazol-4-yl)propan-1-one
N-{1-[3-(2-ethylbutyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]-1-oxopropan-2-yl}propanamide
(3S,4R)-1-(4-ethyl-5-methylthiophene-3-carbonyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
3-{[(2S,5R)-5-(thiomorpholin-4-ylmethyl)oxolan-2-yl]methyl}benzonitrile
2-benzyl-4-[2-(prop-2-yn-1-yloxy)phenyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]-N-(1,3-dimethyl-1H-pyrazol-4-yl)acetamide
N-(1-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
(3S,9aR)-3-[(2S)-butan-2-yl]-8-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]acetamide
2-{1-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]propyl}-2,3-dihydro-1H-isoindol-1-one
N-[3-(2-ethoxyphenyl)propyl]-2-(morpholin-2-yl)acetamide
1-cyclohexyl-4-(oxolane-2-carbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
4-[(4-fluorophenyl)methyl]-1-[(2-hydroxyphenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
7-(2,3-dimethoxyphenyl)-9-methoxy-4-[(4-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[3-(5-methylfuran-2-yl)-5-[4-(4-methylpiperazin-1-yl)phenyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
3-cyclopentyl-N-{[1-(pyridin-2-ylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}propanamide
N-[(1-ethylpiperidin-4-yl)methyl]-4-methyl-1H-imidazole-2-carboxamide
1-(4-{2-methoxy-5-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
1-[(6-hydroxypyrimidin-4-yl)methyl]-3-[3-(4-methylpiperidine-1-carbonyl)phenyl]urea
N-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
4-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]benzoic acid
N-[(5-chloro-2-ethoxyphenyl)methyl]-N,6,6-trimethyl-5-oxothiomorpholine-3-carboxamide
2-methyl-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-1,4-diazepan-5-one
1-{4-[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-1,4-diazepan-1-yl}ethan-1-one
1-[(4aR,8aR)-7-{[4-(difluoromethoxy)phenyl]methyl}-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
N-[(5-methylpyrazin-2-yl)methyl]-2-(naphthalen-2-yloxy)propanamide
1-methyl-4-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
methyl 5-[(cyclohex-3-en-1-ylmethyl)amino]-1-(2-methoxyethyl)-3-(3-methylbutanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
6-(2,5-dimethylfuran-3-yl)-N-(3-methylbutyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
ethyl 2-amino-3-cyano-4-(2-methylphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-6-carboxylate
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)pyridine-3-carboxamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(4-ethylpiperazin-1-yl)acetamide
(3R)-1-[1-(4-fluorophenyl)cyclopropanecarbonyl]-3,4,4-trimethylpyrrolidin-3-ol
1-[(6,7-dimethoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-N-ethylpyrrolidine-3-carboxamide
6-[({[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}amino)methyl]-1,4-oxazepan-6-ol
4-(4-cyclopropanecarbonyl-1,4-diazepan-1-yl)-6-ethyl-N,N-dimethylpyrimidin-2-amine
2-[4-(quinolin-4-ylmethyl)morpholin-3-yl]acetic acid
1-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(1H-imidazol-2-ylmethyl)[2-(1H-indol-1-yl)ethyl]methylamine
4-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-[1-(3-methylphenyl)-1H-imidazol-2-yl]-1-[(2S)-oxolan-2-ylmethyl]-4-phenyl-1H-imidazole