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1-[3-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
N-cyclohexyl-N-methyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
3-(2-methoxyphenyl)-1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]propan-1-one
4-{[3-cyclopentyl-1-(3,4-dimethylphenyl)-1H-1,2,4-triazol-5-yl]methyl}piperazin-2-one
N-[1-(pyrazin-2-yl)propan-2-yl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-methyl-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]-N-[(3-methylpyridin-4-yl)methyl]acetamide
(2S,4R)-N,N-diethyl-4-[2-(4-hydroxyphenyl)acetamido]-1-methylpyrrolidine-2-carboxamide
N-(carbamoylmethyl)-2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-methoxy-5-methyl-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]thiophene-2-carboxamide
2-cyclopentyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-phenylacetamide
5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-3-[2-(methylsulfanyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
4-ethyl-3-{[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(3,4-difluorophenyl)-4-(3-propoxypiperidin-1-yl)piperidine
2-[2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-{1-oxo-1-[3-(pyridin-2-yl)azetidin-1-yl]propan-2-yl}pyrrolidin-2-one
1-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
N-[2-(2-fluorophenyl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-5,6,7,8-tetrahydroquinoline-3-carboxamide
3-(dimethylamino)-N-[1-(3-phenylpropyl)piperidin-3-yl]benzamide
1-[4-(2-hydroxyethyl)piperazin-1-yl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butan-1-one
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-(1H-imidazol-2-ylmethyl)-8-azabicyclo[3.2.1]octane
(2S,4S)-N-ethyl-4-(5-methylthiophene-2-amido)-1-(1,2-oxazole-3-carbonyl)pyrrolidine-2-carboxamide
2-amino-4-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-1,3-thiazole-5-carboxamide
5-[(cyclohexylmethyl)amino]-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(4-chloro-1H-pyrazol-1-yl)-1-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]propan-1-one
8-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-1-[(2-fluorophenyl)methoxy]-1,8-diazaspiro[4.5]decan-2-one
1-(3-chlorophenyl)-4-(1H-indole-5-carbonyl)-5-methylpiperazin-2-one
4-{4-[(5-chloro-2-hydroxyphenyl)methyl]piperazin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
7-(cyclopropylmethyl)-N-ethyl-6-(4-methoxyphenyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(8-fluoroquinoline-2-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
2-{4-[(4-aminopiperidin-1-yl)methyl]phenyl}-6-(2-chlorophenyl)-3,4-dihydropyrimidin-4-one
1-ethyl-3,5-dimethyl-N-[2-(propylsulfanyl)ethyl]-1H-pyrazole-4-carboxamide
8-[(5-methoxy-2-methyl-3-phenyl-1-benzofuran-6-yl)methyl]-1-methyl-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(morpholin-4-yl)-3-{1-[(4-phenylphenyl)methyl]piperidin-4-yl}propan-1-one
2-{4-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
3-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridazine
5-ethyl-1'-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(1-propyl-1H-imidazol-2-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
4-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-1,3-dimethyl-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-1-[(diethylcarbamoyl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-cyclobutyl-6-methyl-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}pyrimidin-2-amine
3-[(2R,3R,6R)-5-[(2-fluorophenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
(2-propoxy-5-{1H-pyrazolo[3,4-b]pyridin-1-yl}phenyl)methanol
N-methyl-N-(1,2-oxazol-3-ylmethyl)-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
methyl 4-[(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-1-oxo-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-5-yl]benzoate
8-[(6-hydroxy-1,4-oxazepan-4-yl)methyl]-3-oxatricyclo[7.3.1.05,13]trideca-1(12),5(13),6,8,10-pentaen-2-one
5-benzyl-4-[1-(2,6-dimethoxypyridine-3-carbonyl)piperidin-3-yl]-2-methylpyrimidine
1-tert-butyl-N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-5-oxopyrrolidine-3-carboxamide
1-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
N-cyclopentyl-N'-(2-phenoxyethyl)butanediamide