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N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-[2-(morpholin-4-yl)propanoyl]piperidine-4-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(pyrazin-2-yl)piperidine-4-carboxamide
(5S,9aS,9bS)-2-(2-phenylethyl)-5-(thiophen-3-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(2S,4S)-N-ethyl-4-(2-methoxy-4-methylbenzamido)-1-(3-methylbut-2-en-1-yl)pyrrolidine-2-carboxamide
2-(dimethylamino)-N-{[4-(hydroxymethyl)phenyl]methyl}-2-(2-methylphenyl)acetamide
ethyl 2-(1-{2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetamido}cyclohexyl)acetate
3-[2-(methylsulfanyl)benzoyl]-N-(2-phenylethyl)piperidine-1-carboxamide
4-(4-fluorophenyl)-5-methyl-2-{5-methyl-4-[4-(piperidin-1-yl)piperidine-1-carbonyl]-1H-pyrazol-1-yl}pyrimidine
{[4-(1H-imidazol-1-yl)phenyl]methyl}(methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-4-(quinolin-4-ylmethyl)-1,4-diazepan-2-one
(4aR,7aS)-1-propyl-4-(1H-pyrazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-4-methyl-2-phenylpyrimidine-5-carboxamide
1-(furan-2-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3-methyl-1H-1,2,4-triazol-5-yl)acetamide
N'-(3-hydroxy-3-phenylpropyl)-N'-methyl-N-(2-methylphenyl)propanediamide
2-{1-[(dimethylcarbamoyl)methyl]pyrrolidin-3-yl}benzoic acid
4-({4-methyl-5-[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
N-[(3R,4R)-1-(4-cyanopyridin-2-yl)-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
ethyl 4-{1-[2-(2,5-dimethoxyphenyl)acetyl]piperidin-3-yl}piperazine-1-carboxylate
N-(2-{7-[(4-phenylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
1-{5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-yl}-1,4-diazepane
N-[2-(4-hydroxyphenyl)ethyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
7-(3-chlorophenyl)-4-(3-methylfuran-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-{3-[benzyl(methyl)amino]piperidin-1-yl}-N,N-dimethylpyrazine-2-carboxamide
N-[2-chloro-5-(diethylcarbamoyl)phenyl]-2-(methylsulfanyl)pyridine-3-carboxamide
N-[1-(2-hydroxyphenyl)ethyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N'-cyclooctyl-N-(piperidin-4-ylmethyl)butanediamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-phenylcyclopropyl)acetamide
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N,5-dimethyl-N-(oxolan-3-yl)-1H-pyrazole-4-carboxamide
dimethyl(3-{2-[1-(1-methyl-1H-imidazole-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
6-{3-cyclopropyl-5-[1-(morpholin-4-yl)ethyl]-1H-1,2,4-triazol-1-yl}-2-methyl-1,3-benzothiazole
4-(cyclopropanesulfonyl)-9-(cyclopropylmethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
N-[2-(dimethylamino)ethyl]-1-[(2-fluorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-5-(methoxymethyl)furan-2-carboxamide
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]propanamide
3-ethoxy-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]propan-1-one
N-methyl-2-[1-(oxolan-3-ylmethyl)piperidin-4-yl]acetamide
5-(4-acetylphenoxymethyl)-N-[2-(2-oxopiperidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
3-{1-[2-(ethylsulfanyl)ethyl]-4-phenyl-1H-imidazol-5-yl}pyridine
1-cyclopentyl-4-({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1,4-diazepane
2-ethyl-1-(propan-2-yl)-4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine
1-methyl-2-phenyl-4-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperazine
3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(6-cyanopyridin-3-yl)-3-[2-(2-methylpropanesulfonyl)ethyl]urea
2-amino-4-{[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}quinazoline-6-carboxylic acid
2-methyl-N-[(2-methylphenyl)(pyridin-4-yl)methyl]-1,3-thiazole-4-carboxamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(4,6-dimethylpyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,3-dimethoxybenzamide