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1-[4-({3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
3-{2-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
2-(pyridin-3-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}pyrimidine-5-carboxamide
5-(3-fluorophenoxymethyl)-N-(2-hydroxy-2-phenylethyl)-1H-pyrazole-3-carboxamide
1-[3-(2-oxopyrrolidin-1-yl)propyl]-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]piperidin-2-one
1-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-4-(thiophen-2-yl)butan-1-one
5-ethyl-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrimidin-2-amine
1-{1-[(4-ethoxyphenyl)methyl]piperidin-3-yl}-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
3-[(3R,4S)-1-(6-chloro-4-methylquinolin-2-yl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
[2-(1H-imidazol-1-yl)-1-phenylethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
[(3R,4R)-1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-methyl-2-(morpholin-4-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-{2-[3-(3-methylphenyl)piperidin-1-yl]-2-oxoethyl}benzamide
N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}-1H-indole-3-carboxamide
N-[4-({1-[2-(4-methoxyphenyl)ethyl]-3-methyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl}methyl)phenyl]acetamide
4-{4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]phenoxy}-N,N-dimethylpiperidine-1-sulfonamide
3-cyclopropyl-4-[2-(4-methoxyphenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(3-acetylphenyl)-3-(piperidin-1-yl)azetidine-1-carboxamide
(1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-[(4-methoxyphenyl)methyl]piperidin-4-yl)methanol
1-[4-(1H-pyrazol-1-yl)benzoyl]-4-(thian-4-yl)piperazine
1-benzyl-5-{[(5-chlorothiophen-2-yl)methyl]amino}-N-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl (1R,3S,3aR,6aS)-3-[4-methoxy-3-(methoxymethyl)phenyl]-1,5-dimethyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-(4-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(3-methylbut-2-en-1-yl)piperazin-2-yl)ethan-1-ol
1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-4-(pyrrolidin-3-yl)piperazine
2-methoxy-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)propanamide
5-chloro-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}thiophene-2-carboxamide
4-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-3-yl]-5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]pyrimidine
(1s,4s)-N-ethyl-4-hydroxy-N-(2-phenoxyethyl)cyclohexane-1-carboxamide
2-[1-(5-chloro-2-methoxyphenyl)-5-(1,2-oxazol-3-yl)-1H-1,2,4-triazol-3-yl]acetamide
2-(4-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
2-{4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]phenyl}acetic acid
4-[3-(1-methylpiperidin-2-yl)propanoyl]-1-(2-phenylethyl)piperazin-2-one
(1S,5R)-6-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,2-dimethyloxane-4-carboxamide
1-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-1,4-diazepane
2-{4-[1-(2-methoxyphenyl)-1H-imidazol-2-yl]phenoxy}acetamide
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-[3-(pyridin-3-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
9-(6-methylpyridine-2-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 4-[4-(5-ethyl-1,2,4-oxadiazol-3-yl)piperazin-1-yl]benzoate
7-(2-hydroxyethyl)-2-(1-methyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-(1-{7-[(2,3-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
2-methyl-5-{[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)propyl]sulfanyl}-1,3,4-thiadiazole
ethyl 4-(3-{[(cyclohexylmethyl)amino]methyl}-6-methylquinolin-2-yl)piperazine-1-carboxylate
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(3,4-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
(3S,4S)-4-(dimethylamino)-1-(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)pyrrolidin-3-ol
5-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]quinoxaline
2-(2,3-dihydro-1H-indol-1-yl)-1-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethan-1-one
2-[1-(4-methoxyphenyl)-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]morpholine
N-[(2S)-1-hydroxy-3-(1H-indol-3-yl)propan-2-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide