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1-(oxolan-3-ylmethyl)-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
3-[4-(5-propyl-1,2-oxazole-3-carbonyl)piperazin-1-yl]-1λ6-thiolane-1,1-dione
1-{2,7-diazaspiro[4.5]decan-2-yl}-2-methoxyethan-1-one
N-[4-(4-fluorophenoxy)phenyl]-7-methyl-2,7-diazaspiro[4.4]nonane-2-carboxamide
2-{4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-benzyl-2-tert-butyl-4-hydroxy-N-[(1R,2R)-2-hydroxycyclohexyl]pyrimidine-5-carboxamide
N-[3-(propan-2-yloxy)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-(cyclopropylmethyl)-2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-methyl-1,3-oxazole-4-carboxamide
7-(cyclohexylmethyl)-2-{[5-(methoxymethyl)furan-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
3-[({[1-(hydroxymethyl)cyclopentyl]methyl}carbamoyl)methyl]-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-ethyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-oxopiperazin-2-yl)-N-methylacetamide
3-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-N-(3,4,5-trifluorophenyl)piperidine-1-carboxamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({[1-(methoxymethyl)cyclopentyl]amino}methyl)piperidin-2-one
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-methyl-N-[2-(morpholin-4-yl)ethyl]azepan-4-amine
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-methyl-1H-imidazole-5-carboxamide
N-[(3R,4S)-1-[3-oxo-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-4-propylpyrrolidin-3-yl]acetamide
[4-(thiomorpholin-4-yl)quinazolin-2-yl]methanol
N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
4-(hydroxymethyl)-1-(2-phenoxybenzoyl)piperidin-4-ol
2-(4-{[methyl(6-methyl-2-phenylpyrimidin-4-yl)amino]methyl}piperidin-1-yl)ethan-1-ol
[(8-methoxyquinolin-5-yl)methyl](methyl){[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
(1R,3S)-3-({2-[2-(propan-2-yloxy)phenyl]ethyl}carbamoyl)cyclopentane-1-carboxylic acid
4-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidine-1-carbonyl}-6-(2-methylpropyl)-1,2-dihydropyrimidin-2-one
2-ethyl-N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)pyrimidine-5-carboxamide
2,3,5,6-tetramethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
1-[4-({4-[(2,4,5-trimethylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
methyl[1-(pyridin-3-yl)ethyl]{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
1-{[2-(difluoromethoxy)phenyl]methyl}-4-(2-methylpropyl)-1,4-diazepan-5-one
N-[(2R,3R)-1'-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
N-[4-(1-ethyl-1H-1,2,4-triazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]cyclopentanecarboxamide
dimethyl({[(3S,4R)-1-(2-phenoxyethyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl})amine
(3aR,6aS)-5-{[4-(cyclopentyloxy)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-methyl-3-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2-dihydroquinolin-2-one
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
[5-(1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1H-1,2,3-triazol-4-yl)furan-2-yl]methanol
N-(1-benzothiophen-2-ylmethyl)-6-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
2-methoxy-2-phenyl-N-[1-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
(2S,4S)-4-amino-N-ethyl-1-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}pyrrolidine-2-carboxamide
N'-(2-tert-butylphenyl)-N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)butanediamide
2,3-dimethyl-N-(thiolan-3-yl)quinoxaline-6-carboxamide
2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-{3-[2-(2-chloro-4-fluorophenyl)-1H-imidazol-1-yl]propyl}-4-methylpiperazine
3-{[7-acetyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl](methyl)amino}-N-methylpropanamide
1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
3-[methyl(1-methylpyrrolidin-3-yl)carbamoyl]benzoic acid
N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-1,2,5-thiadiazole-3-carboxamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(3,4-difluorophenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
3-({[2-(6-methylpyridin-2-yl)ethyl]amino}methyl)pyrrolidin-3-ol
N-methyl-N-(1-methylpyrrolidin-3-yl)-5,6,7,8-tetrahydroquinoline-3-carboxamide