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N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
3-{[6-methyl-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidin-5-yl]formamido}-N-(1,3-thiazol-2-yl)propanamide
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2-methylphenyl)-1,4-diazepane
2-(3-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
(2S)-2-[(5-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carbonyl}pyridin-2-yl)amino]propanamide
4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-N-[3-(methylsulfanyl)phenyl]piperidine-1-carboxamide
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
5-methoxy-2-({3-[5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenol
2-amino-8-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-[2-methyl-3-({[2-(pyridin-3-yloxy)propyl]amino}methyl)-1H-indol-1-yl]acetamide
1-{2-[3-(2-chlorophenoxy)azetidin-1-yl]-2-oxoethyl}-4-phenylpyrrolidin-2-one
3-{[(4aS,8aR)-2-oxo-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-6-yl]methyl}benzonitrile
5-({3-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)-2-methylpyridine
2-{2-[2-(2-ethyl-1-benzofuran-3-yl)-1H-imidazol-1-yl]ethyl}pyrazine
(2-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-1,3-thiazol-4-yl)methanol
3-(benzylsulfanyl)-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]propanamide
(3aR,6aR)-2-[(3-chloro-5-fluorophenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[(3-fluorophenyl)methyl]-1-{[4-(methylsulfanyl)phenyl]methyl}-1,4-diazepan-5-one
2-(2-ethylbutanoyl)-N-(thiophen-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
3-(oxolan-2-yl)-7-[(2,4,6-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
4-[1-(1-benzofuran-2-ylmethyl)pyrrolidin-3-yl]-2-(pyridin-4-yl)pyridine
2-({methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)pyridine-3-carboxylic acid
2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-N-(1H-1,2,4-triazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[2-methyl-6-(2-methylpropyl)pyrimidine-4-carbonyl]pyrrolidin-3-yl]methanol
4-[(2-methylphenyl)methyl]-1-[4-(piperidin-1-yl)benzoyl]-1,4-diazepan-5-one
1-acetyl-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)piperidine-3-carboxamide
1-(2-ethoxypyridine-3-carbonyl)-2-(furan-2-yl)azepane
2-{[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]methyl}-3,4-dihydroquinazolin-4-one
1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2-oxo-3-(pentan-3-yl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-[3-hydroxy-1-(4-methylphenyl)propyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
4-chloro-N-[3-(2-methoxybenzamido)phenyl]-1-methyl-1H-pyrazole-5-carboxamide
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-phenylpiperazine
3-{2-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl}-7-methyl-2,3-dihydro-1H-indol-2-one
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-(3-ethoxypropyl)-1H-pyrazole-4-carboxamide
2-amino-4-(2,5-dimethoxyphenyl)-6-(3,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-cyclohexyl-4-[2-(methylsulfanyl)pyridine-3-carbonyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
5-[2-(benzylamino)pyrimidin-4-yl]-2-ethoxybenzoic acid
4-[4-({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)piperidin-1-yl]-6-methylpyrimidin-2-amine
1-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}-4-(piperidin-1-yl)piperidine
N,2,4-trimethyl-N-{[3-(methylsulfanyl)phenyl]methyl}-1,3-thiazole-5-carboxamide
1-[(2-chloro-6-fluorophenyl)methyl]-1-ethyl-3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)urea
3-{3-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-3-oxopropyl}-3,4-dihydroquinazolin-4-one
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-({4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-decahydro-1,6-naphthyridin-2-one
(2S,4S)-4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-methyl-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
1-[5-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(piperidin-1-yl)propan-2-ol
3-(2-methoxyethyl)-5-(1,2-oxazol-3-yl)-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-5-methyl-1-phenylpiperazin-2-one
5-fluoro-N4,N4-dimethyl-N2-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]pyrimidine-2,4-diamine