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3-(2H-1,3-benzodioxol-5-yl)-1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
3-({4-[(dipropylamino)methyl]phenyl}formamido)-5-methylhexanoic acid
2-methoxy-2-phenyl-N-{1-[1-(pyrimidin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
1-(4-methoxybenzoyl)-4-(1-methyl-1H-pyrazole-4-carbonyl)piperazine
(1R,5S,8S)-8-methoxy-3-(3-methylthiophene-2-carbonyl)-3-azabicyclo[3.2.1]octane
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
4-(pyrrolidin-1-yl)-6-{1-[(1R,2S,3S,4R,5S)-tricyclo[3.2.1.02,4]octane-3-carbonyl]piperidin-4-yl}pyrimidine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(1H-imidazol-4-yl)ethan-1-one
2-(2-methoxypyridin-3-yl)quinoxaline
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2-(2,3,6-trimethylphenoxy)acetamide
6-fluoro-2-({3-[(4-methylpiperazin-1-yl)methyl]piperidin-1-yl}methyl)quinolin-4-ol
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-[(oxolan-3-ylmethyl)sulfamoyl]benzamide
4-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
2-(3-{[2-(8-methylquinolin-5-yl)-1H-imidazol-1-yl]methyl}piperidin-1-yl)ethan-1-ol
N-[(5-ethylpyridin-2-yl)methyl]-N,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-cyclobutanecarbonyl-N-methyl-N-[1-(pyridin-4-yl)ethyl]piperidine-4-carboxamide
dimethyl[3-(2-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}-1H-imidazol-1-yl)propyl]amine
(1S,9S)-11-{[6-chloro-4-(morpholin-4-yl)quinazolin-2-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
N-{2-[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-(2-oxopyrrolidin-1-yl)benzamide
3-({[5-methyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-yl]amino}methyl)-1λ6-thiolane-1,1-dione
1-[(4-chlorophenyl)methyl]-N-(1H-indol-2-ylmethyl)-6-oxopiperidine-3-carboxamide
5-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-1,3,6-trimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1,3-dimethyl-N-[1-(4-methyl-1H-imidazol-2-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-[({3-[(pyridin-3-yl)amino]propyl}amino)methyl]pyrrolidin-3-ol
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methoxyphenyl]-6-methylpyrimidin-2-amine
6-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-N-(2-methoxyethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-{[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
3-fluoro-N-[1-(1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
N-[(1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]acetamide
7-(cyclobutylmethyl)-2-[3-(4-methoxyphenyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-(1-cycloheptylpiperidin-3-yl)-3,5-dimethyl-1,2-oxazole-4-sulfonamide
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-(2-phenylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[4-(3-methoxyphenoxy)phenyl]-3-(oxan-3-ylmethyl)urea
N-cyclopentyl-5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
7-methyl-3-[2-(methylamino)-1,3-thiazole-4-carbonyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
ethyl 3-[(4-fluorophenyl)methyl]-1-(pyridine-4-carbonyl)piperidine-3-carboxylate
1-{3-[1-(5-chloro-2-methoxyphenyl)-3-ethyl-1H-1,2,4-triazol-5-yl]propyl}pyrrolidin-2-one
5-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]pyrazin-2-ol
5-cyclopropyl-N-[2-(diethylamino)ethyl]-N-ethyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carboxamide
1-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyrimidin-4-ylmethyl)acetamide
4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-N-[5-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-(3,5-difluoropyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
3-(2-methylquinolin-4-yl)-3,9-diazaspiro[5.6]dodecan-10-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-(methylamino)acetamide
{4-[(2,4-dimethylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}(pyridin-3-yl)methanol
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]acetamide
methyl 2-{8-[(3-methoxyphenyl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetate