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5-methyl-2-[1-(oxane-2-carbonyl)-4-(pyrrolidin-1-ylmethyl)piperidin-4-yl]pyridine
5-(3-{[4-(3,5-difluorophenyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)pyrimidine
3-[2-(azepan-1-yl)-2-oxoethyl]-4-[(4-ethoxyphenyl)methyl]piperazin-2-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}piperidine-4-carboxamide
2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]-1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-[2-(2-methoxyethoxy)acetyl]-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
3-[(2,4-difluorophenyl)methyl]-1-(pyrimidin-2-yl)piperidine-3-carboxylic acid
ethyl 4-(oxan-2-ylmethyl)-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-4-carboxylate
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[(2,3,4-trifluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl](4-methoxy-4-methylpentan-2-yl)amine
{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propanamide
N-[3-(1,3-oxazol-5-yl)phenyl]-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
2-amino-4-(5-chloro-2,4-dimethoxyphenyl)-6-(pyridin-2-yl)pyridine-3-carbonitrile
2-{4-[(2-methyl-1,3-thiazol-5-yl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-methoxy-1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidine
1-[2-(aminomethyl)piperidin-1-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
2-(3-hydroxyphenyl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2,3-dimethyl-7-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}-1H-indole
3-(furan-2-yl)-1-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}propan-1-one
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-3-[methyl(1-methylpyrrolidin-3-yl)amino]propanamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)cyclohex-3-ene-1-carboxamide
3-{2-oxo-2-[2-(thiophen-2-yl)azetidin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(1-benzyl-1H-imidazol-2-yl)methyl]-1-methyl-3-(trimethyl-1H-pyrazol-4-yl)urea
4-(5-{[(5-chloropyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)-1-cyclohexylpiperazin-2-one
methyl 1-methoxy-8-[2-(methylsulfanyl)benzoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
7-[2-(1H-imidazol-1-yl)propanoyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}(2,1,3-benzoxadiazol-5-ylmethyl)amine
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]propanamide
N-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-1-(thian-4-yl)piperidin-4-amine
5-{[5-({3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)furan-2-yl]sulfanyl}-1H-1,2,4-triazole
6-(2-aminoethyl)-N-(isoquinolin-5-ylmethyl)-N,2-dimethylpyrimidin-4-amine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]pent-4-enamide
2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(5-methyl-1,2-oxazol-3-yl)acetamide
N-tert-butyl-2-(4-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxy)acetamide
3-(benzyloxy)-1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidine
N-[(2-amino-1,3-thiazol-4-yl)methyl]-2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
2,3,5-trimethyl-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N3-[(2,3-dimethoxyphenyl)methyl]-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}propanamide
1-(2-methoxyphenyl)-4-(3-methyl-1H-pyrazole-5-carbonyl)piperazin-2-one
6-methoxy-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{[5-(3-fluoropyridin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
2-[5-cyclopropyl-4-(4-propylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-[2-(trifluoromethyl)phenyl]pyrimidine
1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-2-(3-methylphenoxy)ethan-1-one
(1R,5R)-3-methanesulfonyl-6-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
(1S,2R)-N1-methyl-N1-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-N2-propylcyclohexane-1,2-dicarboxamide
3,5,7-trimethyl-N-(1,4-oxazepan-6-ylmethyl)-1H-indole-2-carboxamide