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2-[(3-fluorophenyl)methyl]-4-[4-(2-methylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-methyl-1H-pyrazole-4-carboxamide
4-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazine-1-carbonyl)morpholine
2-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]methyl}-6-methylpyridine
N-(2-ethoxypropyl)-N,5,7-trimethylpyrido[2,3-d]pyrimidin-4-amine
1-(3-{[3-(aminomethyl)pyrrolidin-1-yl]methyl}-2,4,6-trimethylphenyl)ethan-1-one
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrazole-4-carboxamide
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-[3-(3-ethylphenoxy)propyl]-N-methyloxane-4-carboxamide
1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3-(2-methoxybenzoyl)piperidine
(4aS,8aR)-1-(3-methoxypropyl)-6-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
(1R,5S)-6-{3-[(1-cyclopentylpiperidin-4-yl)oxy]benzoyl}-6-azabicyclo[3.2.1]octane
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[(2-fluorophenyl)methyl]piperidine
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(oxolan-2-ylmethyl)acetamide
ethyl 3-benzyl-1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidine-3-carboxylate
5-ethyl-N-[2-(pyrrolidin-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-[(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridin-2-amine
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[1-(2-methoxyphenyl)ethyl]methylamine
5-methanesulfonyl-2-(2-methylpropyl)-4-(piperidin-3-yl)pyrimidine
1-ethyl-N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1H-pyrazole-3-carboxamide
3-{[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
(3aR,6aR)-2-methyl-5-[4-(piperidin-1-yl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
[1-(3-fluoro-4-methoxybenzoyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
2-[(2-methoxyethyl)(methyl)amino]-N-[3-(2-phenylacetamido)phenyl]acetamide
3-(2-{5-[5-(hydroxymethyl)furan-2-yl]-4-phenyl-1H-imidazol-1-yl}ethyl)-1,3-oxazinan-2-one
3-chloro-4-({1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
7-{3-[(dimethylamino)methyl]benzoyl}-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-(2-methoxy-5-{[methyl(oxan-4-ylmethyl)amino]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
4-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperazin-1-yl}-2-(2-methoxyethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[(2,6-difluorophenyl)methyl]-2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[5-(methoxymethyl)furan-2-carbonyl]piperidine
N,N-diethyl-2-(4-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)acetamide
2-[5-(4-cyanooxan-4-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl]acetamide
1-methyl-4-{1-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]pyrrolidin-3-yl}piperazine
2-{1-[(4-methylphenyl)methyl]-4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
4-{5-[(2E)-3-phenylprop-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}morpholine
N-(2-methoxyethyl)-6-[3-(methoxymethyl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-{[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}-2-(thiophen-3-yl)acetic acid
5-{1-[(5-chlorothiophen-2-yl)methyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
3-(2,4-difluorophenyl)-1-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidin-1-yl]propan-1-one
3-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,5-dichlorophenyl)urea
2-methyl-3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]pyridine
N3-(3-methylbutyl)-N5-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(3aR,7aS)-2-({3-methoxy-2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
3-{1-[2-(3-hydroxyphenyl)acetyl]piperidin-3-yl}propanamide
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-(pyridin-3-ylmethyl)acetamide