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2-(4-{3-[(1R,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]pyridin-2-yl}piperazin-1-yl)-N-ethylacetamide
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
(2S)-N-[2,3-dimethyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-2-(3-ethyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carboxamide
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
8-(6-methylpyridine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[2-(4-chlorophenyl)ethyl]-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-methoxy-N-[2-(5-methylfuran-2-yl)ethyl]-4-[(1-methylpiperidin-4-yl)oxy]benzamide
N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-{[3-(3-ethoxyphenoxy)-4-methoxyphenyl]methyl}pyrrolidine
1-[4-(2-methoxybenzoyl)piperazin-1-yl]-2-propoxyethan-1-one
2-[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]-1-methyl-1H-1,3-benzodiazole
2-{3-cyclopropyl-5-[(oxolan-2-ylmethoxy)methyl]-1H-1,2,4-triazol-1-yl}pyridine
N-(2-methylpropyl)-1-[1-(quinolin-4-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
6-[1-(4-chlorophenyl)cyclobutanecarbonyl]-N-[2-(cyclohex-1-en-1-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-1-[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]propan-1-one
1'-(4-aminopyrimidin-2-yl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
6-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]pyridine-3-carboxamide
1-[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]-3-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]urea
[(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl][(3-fluorophenyl)methyl]methylamine
N-tert-butyl-2-{[(3-hydroxy-2-oxo-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]amino}acetamide
N2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-N4-ethylpyrimidine-2,4-diamine
1-[(5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}furan-2-yl)methyl]pyrrolidine
2-chloro-3-({[2-(dimethylamino)ethyl](thiophen-3-ylmethyl)amino}methyl)-6-methoxyphenol
4-cyclopentyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrimidin-2-amine
1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
4-(1-methyl-1H-imidazol-2-yl)-1-[(2,3,5,6-tetrafluoro-4-methoxyphenyl)methyl]piperidine
N,N-dimethyl-2-{[(2-methyloxolan-2-yl)formamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
[(1-{1-[(2-chloro-4-fluorophenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]urea
3-chloro-5-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
1-ethyl-4-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}piperazine-2,3-dione
1-benzyl-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrrolidin-3-amine
6-fluoro-4-hydroxy-N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)quinoline-3-carboxamide
(4aS,7aR)-1-[5-(methoxymethyl)furan-2-carbonyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}cyclopropan-1-amine
(2S,4S)-N-ethyl-4-{[(3-methylphenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-[2-(pyridin-2-yl)ethyl]pyrimidin-2-amine
(3S,4S)-1-(6-methoxypyrimidin-4-yl)-4-(naphthalen-2-yl)piperidin-3-ol
4-(1H-1,3-benzodiazol-2-yl)-1-cyclohexyl-3-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-cyclohexyl-4-[(2S)-5-oxopyrrolidine-2-carbonyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-cyclobutyl-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]ethan-1-one
3-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-1,3-thiazolidine
{5-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]furan-2-yl}methanol
N-(2,3-dimethylphenyl)-2-{[(4-phenyloxan-4-yl)methyl]amino}acetamide
6-methyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydroquinolin-2-one
2-{[(3R,5S)-1-[(4-ethoxyphenyl)methyl]-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]pyrrolidin-3-yl]sulfanyl}-1H-1,3-benzodiazole
2-ethyl-4-phenyl-9-[2-(propan-2-yloxy)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
(3R)-1-{[4-phenyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-3-ol
2-{2-[(1-carbamoylpiperidin-3-yl)formamido]ethyl}-4-methyl-1,3-thiazole-5-carboxylic acid
2-(4-{[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)-1-(morpholin-4-yl)ethan-1-one
1-[benzyl(methyl)amino]-3-[5-({[(4,6-dimethylpyrimidin-2-yl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol