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N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2,3-dihydro-1H-inden-2-amine
4-(3,5-dimethoxyphenyl)-2-methyl-6-(propan-2-yl)pyrimidine
2-[5-(7-chloro-1-methyl-1H-indole-2-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
4-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
1-[(4aS,8aS)-4a-hydroxy-7-[(1-methyl-1H-imidazol-2-yl)methyl]-decahydro-2,7-naphthyridin-2-yl]-3-(methylsulfanyl)propan-1-one
(2S,4R)-N,N-diethyl-1-(2-methylpropyl)-4-(2-oxo-2-phenylacetamido)pyrrolidine-2-carboxamide
4-(2-{4-[(5-cyclopentylthiophen-2-yl)methyl]piperazin-1-yl}ethyl)morpholine
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-(propan-2-yl)acetamide
1-cyclopropyl-5-({3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)-1H-imidazole
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-2-methoxypyridine-3-carboxamide
2-(4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperazin-1-yl)benzonitrile
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(5-methylfuran-2-yl)ethyl]acetamide
N-phenyl-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrimidin-2-amine
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-methyl-2-(thiophen-2-ylformamido)propanamide
4-(1-methylpiperidin-4-yl)-7-(morpholin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyridine-3-carboxamide
3-[(3-hydroxyazetidin-1-yl)sulfonyl]-N-[3-(pyridin-3-yl)propyl]benzamide
(3S,4S)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrrolidin-3-ol
3-methyl-6-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridazine
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-hydroxy-2-(4-methoxyphenyl)ethan-1-one
1-[(3S,4R)-1-[(3,4-dimethoxyphenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
7-(2-cyclohexylethyl)-2-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}-2,7-diazaspiro[4.5]decane
2-[3-(3-hydroxy-3-methylbutyl)benzoyl]-1,2,3,4-tetrahydroisoquinolin-5-ol
phenyl({1-[1-(quinolin-3-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl})methanol
ethyl 4-{[2-(dimethyl-1,3-thiazol-2-yl)ethyl]amino}piperidine-1-carboxylate
3-({[(3-chlorophenyl)methyl]amino}methyl)-1-(2-cyclohexylethyl)-3-hydroxypiperidin-2-one
2-{3-[4-(cyclopropylmethoxy)phenyl]phenoxy}acetamide
(2R,6R)-4-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(thiophene-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N2-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-N1-(pyridin-3-yl)ethane-1,2-diamine
1-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-4-(prop-2-en-1-yl)-1,4-diazepan-5-one
N-(1-{7-[(2,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
(4aS,7aR)-1-[(4-chloro-3-fluorophenyl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-hydroxy-N-methyl-N-[3-(oxolan-2-yl)propyl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-[(2R,3R)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
N-[4-(4-{[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}piperidin-1-yl)phenyl]benzenesulfonamide
5-(2-methylpropyl)-1'-(4-methylpyrimidin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(4-fluorophenoxy)ethan-1-one
3-(5-ethylpyrimidin-2-yl)-7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecane
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
3-(2-amino-1,3-thiazol-4-yl)-N-[2-(4-fluorobenzenesulfonyl)ethyl]propanamide
2-cyclobutyl-5-fluoro-1-[1-(oxolane-2-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-benzyl-4-(1-ethyl-1H-imidazol-2-yl)-N-methylpiperidine-1-sulfonamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-1-methyl-1H-pyrazole-5-carboxamide
4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-(2-propyl-2H-1,2,3-triazol-4-yl)-2-[4-(thiophen-3-yl)-1H-pyrazol-1-yl]acetamide
1-[3-(4-methyl-1,4-diazepan-1-yl)propanoyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
4-{3-[3-(methoxymethyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
2-(dimethylamino)-4-methyl-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
4-cyclopentyl-3-(2,2-dimethylcyclopropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one