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N-methyl-N-(oxolan-2-ylmethyl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
3-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-5-phenyl-1,2,4-oxadiazole
(1R,3S)-3-(2-aminoethoxy)-7-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-7-azaspiro[3.5]nonan-1-ol
5-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-2-(3-phenylpropyl)-1,3-benzoxazole
5-(6-ethoxypyridazin-3-yl)-1,2,3,4-tetrahydroisoquinoline
(3R,4R)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-3-ol
5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methoxyphenyl]-2,4-dimethoxypyrimidine
6-{[(2,2-dimethylpropyl)(methyl)amino]methyl}-N-(1,4-dioxan-2-ylmethyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
(2S,4S)-4-amino-1-(1-benzofuran-2-sulfonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(3,6-dimethylpyrazin-2-yl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylic acid
7-chloro-N-ethyl-3,5-dimethyl-N-(pyridin-4-ylmethyl)-1-benzofuran-2-carboxamide
1-(2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzoyl)azocane
3-(4-phenyl-1H-pyrazol-5-yl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
2,8-dimethyl-3-[4-(thian-4-yl)piperazine-1-carbonyl]quinoline
4-(4-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)benzoic acid
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-4-(4-methylphenoxy)piperidine-4-carboxamide
1-(1-methylpiperidin-4-yl)-4-[3-(3-methylpiperidine-1-carbonyl)phenoxy]piperidine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
4-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-2-(piperidin-1-ylmethyl)-1,4-oxazepane
1-[(3R,4S)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-3-(thiophen-3-yl)propan-1-one
2-(2,5-dimethylfuran-3-carbonyl)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
1-cycloheptanecarbonyl-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
2-(3-fluorophenyl)-5-(4,4,4-trifluorobutyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
3-{1-[2-(2,4-dichlorophenoxy)acetyl]piperidin-4-yl}-1,3-oxazolidin-2-one
N-[(3,4-difluorophenyl)methyl]-3-[1-(pyrazin-2-yl)piperidin-3-yl]propanamide
N-[2-(4-{[cyclohexyl(methyl)amino]methyl}phenoxy)propyl]-2-(1H-pyrazol-1-yl)acetamide
2-[4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
(4S)-1-(1,4-dimethyl-1H-indole-2-carbonyl)-3,3,4-trimethylpiperidin-4-ol
2-amino-1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
methyl 2-({[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)acetate
8-(1,3-benzothiazole-6-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
6-[3-(3,3-diphenylpiperidin-1-yl)-3-oxopropyl]-2,3,4,5-tetrahydropyridazin-3-one
(4aS,8aR)-6-(3-chlorobenzoyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
7-[4-(pyridin-3-yl)pyrimidin-2-yl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-(5-acetylthiophen-3-yl)-1-[3-(aminomethyl)pyrrolidin-1-yl]ethan-1-one
1-[2-(4-methoxyphenoxy)ethyl]-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
2-methyl-6-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)pyrimidin-4-ol
ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]{[(2R,5S)-5-[(6-methylpyridin-3-yl)methyl]oxolan-2-yl]methyl}amine
N5-benzyl-1-cyclopropyl-N3-methyl-N3-(naphthalen-1-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-1-[4-(trifluoromethyl)phenyl]urea
2-(4-methylpentyl)-4-(piperidine-1-sulfonyl)morpholine
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[6-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]propanoic acid
methyl 2-methoxy-4-(3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamido)benzoate
N-[2-(propan-2-yl)-1H-1,3-benzodiazol-5-yl]-4-(pyridin-4-yl)piperidine-1-carboxamide
5-{1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-1,2,3-triazol-4-yl}pyrimidine
2-{[(1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
2-(5-acetylthiophen-3-yl)-N-(naphthalen-1-ylmethyl)acetamide
7-(4-chlorophenyl)-2-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-phenyl-5-[(2,3,4-trimethoxyphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine