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3-[(3R,4S)-1-[(3-fluoro-2-methylphenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
1-(3-fluorophenyl)-3-{1-[1-(1-methylazepane-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl](quinolin-2-ylmethyl)amine
2-(4-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperazin-1-yl)pyridine-3-carboxamide
2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)-1-(1,4-oxazepan-4-yl)ethan-1-one
1-[(3-fluorophenyl)methyl]-4-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperazin-2-one
1-cyclopropyl-3-{2-[2-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
(4aR,8aS)-1-[(4-fluorophenyl)methyl]-6-(thiophen-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
4-{[5-(dimethylcarbamoyl)furan-2-yl]methoxy}-2-hydroxy-5-(1-methyl-1H-pyrazol-4-yl)benzoic acid
(2S,4R)-N-methyl-4-[(pentan-3-yl)amino]-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
2-(2-methylpropanoyl)-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2,5-dimethyl-1,3-thiazole-4-carboxamide
1-(3-methylbut-2-en-1-yl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
methyl 1-[(3R,5S)-5-{[2-(4-fluorophenyl)ethyl]carbamoyl}-1-(quinolin-4-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-[1-(1H-imidazol-1-yl)butan-2-yl]-3-{5-[(4-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}urea
(3R,4R)-1-[(3,7-dimethyl-1H-indol-2-yl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
2-(4-{4-[(2,3-dihydro-1H-inden-2-yl)amino]piperidin-1-yl}phenyl)-N-[2-(2-methoxyphenyl)ethyl]acetamide
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]furan-2-carboxamide
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
3-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-5,6-dimethyl-1,2-dihydropyridin-2-one
2-[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]-1-(oxan-3-yl)-1H-imidazole
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[(2-fluorophenyl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-oxopiperidine-3-carboxamide
1'-[(4-chlorophenyl)methyl]-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
8-(6-methylpyridazin-3-yl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-butyl-N-methyl-3-({[1-(pyridin-3-yl)propan-2-yl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
methyl 4-({4-[(2-methylphenyl)methyl]-5-oxo-1,4-diazepan-1-yl}methyl)benzoate
2,6-dimethoxy-3-{5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyridine
(4S)-3-{2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-oxoethyl}-4-phenyl-1,3-oxazolidin-2-one
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)benzamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
(3S,4R)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
ethyl 1-(3-cyclopropyl-1H-pyrazole-5-amido)piperidine-3-carboxylate
N-methyl-3-(N-methylmethanesulfonamido)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]propanamide
N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)-1-azabicyclo[2.2.2]octan-3-amine
4-({[6-(2-aminoethyl)pyrimidin-4-yl]amino}methyl)-1,2-dihydrophthalazin-1-one
3-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydroquinolin-2-one
1-(naphthalen-2-ylmethyl)-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-[2-(1H-pyrrol-1-yl)ethyl]piperazine
(1R,5R)-6-[3-(4-hydroxyphenyl)propanoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-[4-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-3-carboxamide
1-tert-butyl-4-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}pyrrolidin-2-one
4-benzyl-3-{1-[4-methyl-6-(methylamino)pyrimidin-2-yl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}-4,6-dimethylpyrimidine
6-[(1H-imidazol-2-ylmethyl)(methyl)amino]-N-methyl-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
N-cycloheptyl-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
[1-(pyridin-3-yl)propan-2-yl](2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)amine