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4-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,4-diazepane-1-carbaldehyde
(1S,5R)-3-benzyl-6-[2-(2-methoxyphenoxy)ethyl]-3,6-diazabicyclo[3.2.2]nonane
1-(1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazol-3-yl)ethan-1-one
3-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)urea
2-[(3,5-difluorophenyl)methyl]-N,N-dimethyl-3-oxo-2,8-diazaspiro[4.5]decane-8-sulfonamide
4-phenoxy-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
3-(dimethylsulfamoyl)-5-[(furan-2-ylmethyl)amino]-N-methyl-N-(1,3-thiazol-2-ylmethyl)benzamide
4-methoxy-N-{[1-(pyridine-3-carbonyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
4-ethyl-1-methyl-3-({1-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-phenyl-1-(2-{[(3,4,5-trimethoxyphenyl)methyl]amino}ethyl)-1H-1,2,3-triazole-4-carboxamide
(4aR,8aS)-6-(furan-2-carbonyl)-1-(4-methoxybenzoyl)-decahydro-1,6-naphthyridine
1-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
N-[(3S,4R)-1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
methyl 5-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-3-(4-methoxybenzamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[2-(methylsulfanyl)ethyl]benzamide
N'-cyclopentyl-N,N-dimethyl-N'-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)butanediamide
4-methoxy-N-[(5-methyl-1,2-oxazol-3-yl)methyl]benzamide
(4aR,8aS)-6-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-(3-ethoxypropyl)-decahydro-1,6-naphthyridin-2-one
N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(4-phenylphenyl)acetamide
3-methoxy-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)propanamide
[2-ethoxy-5-(4-phenyl-1H-imidazol-5-yl)phenyl]methanol
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-butyl-2-(1,4-dimethylpiperazin-2-yl)-N-(3-phenylprop-2-yn-1-yl)acetamide
5-({2-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}sulfanyl)-1H-1,2,3-triazole
1-ethyl-N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(3E)-pent-3-enoyl]pyrrolidin-3-yl]-1H-pyrazole-4-carboxamide
N-(1,3-benzoxazol-2-ylmethyl)-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
4-[2-(methylsulfanyl)ethyl]-1-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
9-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
3-phenyl-1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}pyrrolidin-3-ol
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(2,2,3,3-tetramethylcyclopropanecarbonyl)pyrrolidin-3-yl]methanol
2-{2-[1-(6-methylpyridine-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
5-{[(4-fluorophenyl)methyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-3-phenylpyrrolidin-3-ol
8-(2,6-diaminopyrimidin-4-yl)-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]ethan-1-one
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-ylmethyl)acetamide
N-ethyl-2-{4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperazin-1-yl}acetamide
1-[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]-4-phenylbutan-1-one
3-[2-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-hydroxyethyl]phenol
2-[(5-methylpyrazin-2-yl)methyl]-8-(6-methylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
4-(hydroxymethyl)-3-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3-oxazolidin-2-one
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}({[2-(trifluoromethyl)phenyl]methyl})amine
1-[(3-chlorophenyl)methyl]-4-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
{[2-(difluoromethoxy)phenyl]methyl}({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
1-[(5-chlorothiophen-2-yl)sulfonyl]-3-(4-methoxy-2-methylbenzoyl)piperidine
(2R)-2-methyl-1-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)piperazine
2-amino-6-benzoyl-4-(cyclohex-3-en-1-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-[(2-hydroxyphenyl)methyl]-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-3-(1-methylpiperidin-2-yl)propanamide
3-cyclopropyl-N-(6-methylpyridin-3-yl)-1H-pyrazole-5-carboxamide