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[2-(2-methoxyquinolin-3-yl)-1,3-thiazol-4-yl]methanol
4-sulfamoyl-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]benzamide
N-methyl-4-(2-methyl-1H-imidazol-1-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}butanamide
4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1-methyl-2-phenylpiperazine
N-cyclohexyl-N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]acetamide
(1S,5R)-6-(cyclobutylmethyl)-3-{[2-(ethylamino)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-methoxyethyl)-3-{[2-(pyrazin-2-yl)ethyl]sulfamoyl}benzamide
methyl 3-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}benzoate
methyl 4-({1-methoxy-2-oxo-1,8-diazaspiro[4.5]decan-8-yl}methyl)benzoate
(3S,4S)-4-(4-fluorophenyl)-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-ol
2-{1-[(3-chloro-4-methoxyphenyl)methyl]pyrrolidin-2-yl}-1,3-thiazole
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)acetamide
8-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]quinoline
7-(3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
[3-(2-phenoxyethyl)-1-(4,4,4-trifluorobutyl)piperidin-3-yl]methanol
2-(2,5-dimethoxyphenyl)-2-{methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}acetic acid
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N,N-bis(2-methoxyethyl)pyridin-2-amine
1-(3-chloro-4-hydroxybenzoyl)-4-hydroxypiperidine-4-carboxylic acid
2-{[4-(4-benzyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]methyl}phenol
3-[2-(2,6-difluorophenyl)ethyl]-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}-4-(pyridin-4-yl)piperazine
5-(2,4,6-trimethylphenyl)pyrazin-2-amine
N-(1-{7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)furan-2-carboxamide
1-[2-methoxy-5-({[2-(pyrazin-2-yl)ethyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-5-[(methylsulfanyl)methyl]furan-2-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-(3-methoxy-2,2-dimethylpropyl)-5-methylpiperidin-2-one
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-(1H-imidazol-1-yl)benzamide
3-fluoro-N-{1-[1-(quinolin-8-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-methyl-3-{[3-(4-methylphenoxymethyl)piperidin-1-yl]methyl}pyridin-2-amine
2-(piperidin-1-yl)-N-[2-(thiophen-2-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
4-{2-methoxy-5-[3-methyl-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]phenyl}morpholine
2-[4-(4-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-6-methylpyridine-3-carbonitrile
3-(1-butyl-1H-imidazol-2-yl)-1-(2-methyl-1-benzofuran-5-carbonyl)piperidine
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-[3-(1H-pyrazol-1-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-({[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}methyl)-3,4-dihydroquinazolin-4-one
1-{[3-(cyclopentyloxy)phenyl]methyl}-3-(pyrrolidin-1-yl)piperidine
1-cyclopropanecarbonyl-N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}piperidine-4-carboxamide
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}ethan-1-one
methyl[(2-methyl-1,3-thiazol-4-yl)methyl]{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}amine
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-[(methylsulfanyl)methyl]-4-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]-1,3-thiazole
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-{[7-methoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}-N-(3-methoxypropyl)-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
(1R,7S)-3-tert-butyl-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
5-methyl-1-[4-(pyridin-3-yl)pyrimidin-2-yl]-N-[3-(pyridin-3-yloxy)propyl]-1H-pyrazole-4-carboxamide
1,6-dimethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-benzyl-1-cyclopropyl-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
N4-(1,4-dioxan-2-ylmethyl)-N2,N2,N4,5,6-pentamethylpyrimidine-2,4-diamine
N-{2-[4-(4-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}benzamide