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3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
4-methyl-2-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl}-1H-1,3-benzodiazole
N-[3-(4-hydroxypiperidin-1-yl)propyl]-2,2-dimethylpropanamide
N-{[(3R,4R)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}-2,3,5,6-tetramethylbenzamide
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(3R,4S)-4-{4-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-1,4-diazepan-1-yl}oxolan-3-ol
9-[3-(pyridine-2-carbonyl)piperidin-1-yl]-3-azaspiro[5.5]undecane
N-({3-[2-(2,4-dimethylphenoxy)ethyl]phenyl}methyl)acetamide
1-{3-[(4,4-difluoropiperidin-1-yl)methyl]phenoxy}-3-(morpholin-4-yl)propan-2-ol
1-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-(4-methylpiperazine-1-carbonyl)pyrazin-2-amine
2-(dimethylamino)-2-(3-methylphenyl)-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}ethan-1-one
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
2-[(3,5-difluorophenyl)methyl]-8-(2-hydroxypropyl)-2,8-diazaspiro[4.5]decan-3-one
2-methyl-6-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1,3-benzothiazole
N-({7-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-methoxybenzamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-methyl-3-(5-methyl-1,3,4-thiadiazol-2-yl)urea
1-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-1,2,4-triazol-1-yl)propan-1-one
1-(2-{1-[4-(3-fluorophenyl)benzoyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
5-{[(6-cyclopropylpyrimidin-4-yl)amino]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-methyl-4-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-1-(2-methylpropyl)piperazin-2-one
4-{[2-(pyridin-2-yl)-1H-imidazol-1-yl]methyl}benzene-1-sulfonamide
1-cyclopentyl-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-6-oxopiperidine-3-carboxamide
3-(cyclopentylsulfamoyl)-5-(4-methyl-1H-pyrazol-1-yl)benzoic acid
N-cyclohexyl-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
N-{[5-(4-fluorophenyl)furan-2-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
4-(1-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)pyridine
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-({[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)piperidin-2-one
7-fluoro-3-methyl-N-(quinolin-2-ylmethyl)-1-benzofuran-2-carboxamide
N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-N5-{[2-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
3-(1,3-dimethyl-1H-pyrazol-4-yl)-1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]urea
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3-benzotriazole-5-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(4-methylpyrimidine-5-carbonyl)piperidin-3-ol
9-oxo-N-propyl-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carboxamide
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-methylbutan-1-one
3-(1H-1,3-benzodiazol-1-yl)-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylpropanamide
[2-(diethylamino)ethyl](methyl){[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
(2-{7-[methyl(propan-2-yl)sulfamoyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}-2-oxoethyl)urea
N-[(5-chloro-2-methoxyphenyl)methyl]-1-(2-methoxyacetyl)-N-methylpiperidine-4-carboxamide
4-(3,4-dimethoxyphenyl)-3-[1-(morpholin-4-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-[(1r,4r)-4-hydroxycyclohexyl]acetamide
5,6-dimethyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyrimidin-4-amine
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-ethyl-3-methyl-1H-pyrazole-5-carboxamide
methyl 2-{[(3-fluorophenyl)methyl]sulfamoyl}-6-(2-methylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[2-(ethanesulfinyl)ethyl]-3-(propan-2-yl)-1H-1,2,4-triazole
N-methyl-N-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]acetamide
(2-{5-[(4-methylpiperazin-1-yl)methyl]pyridin-2-yl}phenyl)methanol
2-amino-4-(oxolan-3-yl)-6-(1-propyl-1H-1,2,3-benzotriazol-5-yl)pyridine-3-carbonitrile